An efficient synthesis of cyclic RGD peptides as antithrombotic agents

被引：7

作者：

Zhang, LH

Pesti, JA

Costello, TD

Sheeran, PJ

Uyeda, R

Ma, P

Kauffman, GS

Ward, R

McMillan, JL

机构：

[1] DuPont Merck Pharmaceutical Company, Deepwater

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1996年 / 61卷 / 15期

关键词：

D O I：

10.1021/jo9603284

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：5180 / 5185

页数：6

共 21 条

[1] STRUCTURAL STUDIES OF A FAMILY OF HIGH-AFFINITY LIGANDS FOR GPIIB/IIIA [J].

BACH, AC ;

EYERMANN, CJ ;

GROSS, JD ;

BOWER, MJ ;

HARLOW, RL ;

WEBER, PC ;

DEGRADO, WF .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1994, 116 (08) :3207-3219

[2] CYCLIC RGD PEPTIDE ANALOGS AS ANTIPLATELET ANTITHROMBOTICS [J].

BARKER, PL ;

BULLENS, S ;

BUNTING, S ;

BURDICK, DJ ;

CHAN, KS ;

DEISHER, T ;

EIGENBROT, C ;

GADEK, TR ;

GANTZOS, R ;

LIPARI, MT ;

MUIR, CD ;

NAPIER, MA ;

PITTI, RM ;

PADUA, A ;

QUAN, C ;

STANLEY, M ;

STRUBLE, M ;

TOM, JYK ;

BURNIER, JP .

JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (11) :2040-2048

[3]

BODANSZKY M, 1984, PRINCIPLES PEPTIDE S, V16, P137

[4]

Bodanszky M., 1993, PRINCIPLES PEPTIDE S, V2nd

[5]

Bodanszky M., 1984, PRACTICE PEPTIDE SYN

[6] A MURINE MONOCLONAL-ANTIBODY THAT COMPLETELY BLOCKS THE BINDING OF FIBRINOGEN TO PLATELETS PRODUCES A THROMBASTHENIC-LIKE STATE IN NORMAL PLATELETS AND BINDS TO GLYCOPROTEINS-IIB AND OR GLYCOPROTEIN-IIIA [J].

COLLER, BS ;

PEERSCHKE, EI ;

SCUDDER, LE ;

SULLIVAN, CA .

JOURNAL OF CLINICAL INVESTIGATION, 1983, 72 (01) :325-338

[7] O-BENZOTRIAZOLYL-N,N,N',N'-TETRAMETHYLURONIUM HEXAFLUOROPHOSPHATE AS COUPLING REAGENT FOR THE SYNTHESIS OF PEPTIDES OF BIOLOGICAL INTEREST [J].

DOURTOGLOU, V ;

GROSS, B ;

LAMBROPOULOU, V ;

ZIOUDROU, C .

SYNTHESIS-STUTTGART, 1984, (07) :572-574

[8] TRIMETHYLSILYL TRIFLUOROMETHANESULFONATE AS A USEFUL DEPROTECTING REAGENT IN BOTH SOLUTION AND SOLID-PHASE PEPTIDE SYNTHESES [J].

FUJII, N ;

OTAKA, A ;

IKEMURA, O ;

AKAJI, K ;

FUNAKOSHI, S ;

HAYASHI, Y ;

KURODA, Y ;

YAJIMA, H .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1987, (04) :274-275

[9]

GOULD RJ, 1990, P SOC EXP BIOL MED, V195, P168, DOI 10.3181/00379727-195-43129B

[10] CYCLO(DIPEPTIDE)S AS LOW-MOLECULAR-MASS GELLING AGENTS TO HARDEN ORGANIC FLUIDS [J].

HANABUSA, K ;

MATSUMOTO, Y ;

MIKI, T ;

KOYAMA, T ;

SHIRAI, H .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1994, (11) :1401-1402

← 1 2 3 →