Vilsmeier-Haack reaction: A manifest protocol to synthesise bisquinoline

被引：0
作者：
Makhanya, T. R. [2 ]
Pitchai, P. [1 ]
Gengan, R. M. [2 ]
Mohan, P. S. [3 ]
机构：
[1] Govt Arts Coll, PG & Res Dept Chem, Kumbakonam 612001, India
[2] Durban Univ Technol, Dept Chem, ML Sultan Campus, ZA-4001 Durban, South Africa
[3] Bharathiar Univ, Dept Chem, Sch Chem Sci, Coimbatore 641046, Tamil Nadu, India
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2016年 / 55卷 / 04期
基金：
新加坡国家研究基金会;
关键词：
Bisquinolines; Claisen condensation; Vilsmeier-Haack reaction; Schiff base; MICROWAVE-ASSISTED SYNTHESIS; ANTIMALARIALS;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Synthesis of bisquinolines from methyl anthranilate and ethyl acetbacetate is described. This synthesis has been accomplished in three steps. Vilsmeier-Haack reaction is used as a key tool to assemble bisquinoline. Microwave heating during each step of the reaction gives high yield of products in short reaction times.
引用
收藏
页码：517 / 521
页数：5
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