Synthesis and biological activity of certain 1-substituted-4-benzylidene-2-phenyl-5-imidazolones

被引：0

作者：

Arief, MMH ^{[1
]}

机构：

[1] Benha Univ, Fac Sci, Dept Chem, Benha, Egypt

来源：

REVUE ROUMAINE DE CHIMIE | 1999年 / 44卷 / 02期

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A novel series of 1-substituted-4-benzylidene-2-phenyl-5-imidazolone derivatives were synthesized for their potential biological activity. The synthesis involved the base and acid catalyzed reactions of azide 3 and/or acid chloride 2. Compounds 5c and 5d were easily cyclized to give 1,3,4-oxadiazole derivatives 6a and 6b. Representative examples for internal Friedel-Crafts and [4 + 2] cycloaddition were also investigated.

引用

页码：173 / 179

页数：7

共 10 条

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