ONE-POT SYNTHESIS OF 6-SUBSTITUTED AMINO-2,4-DIAMINOPYRIMIDINE DERIVATIVES USING KETENE DITHIOACETALS WITH AMINES AND GUANIDINE CARBONATE

被引：5

作者：

Hirose, Miki ^{[1
]}

Hagimori, Masayori ^{[2
]}

Shigemitsu, Yasuhiro ^{[3
]}

Mizuyama, Naoko ^{[4
]}

Wang, Bo-Cheng ^{[5
]}

Tominaga, Yoshinori ^{[1
]}

机构：

[1] Nagasaki Univ, Fac Environm Studies, Nagasaki 8528521, Japan

[2] Nagasaki Int Univ, Fac Pharmaceut Sci, Nagasaki 8593298, Japan

[3] Technol Ctr Nagasaki, Nagasaki 8560026, Japan

[4] Saga Univ Hosp, Dept Pharm, Saga 8498521, Japan

[5] Tamkang Univ, Dept Chem, Tamsui 251, Taiwan

来源：

HETEROCYCLES | 2009年 / 78卷 / 04期

关键词：

Pyrimidine; Solid State; Fluorescence; Ketene Dithioacetal; Organic Electron Luminescent; PYRIDAZINES;

D O I：

10.3987/COM-08-11587

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

6-Substituted amino-2,4-diaminopyrimidine derivatives were prepared by one-pot synthesis using ketene dithioacetals, amine compounds, and guanidine carbonate in pyridine. These pyrimidine products displayed blue fluorescence in the solid state.

引用

页码：899 / 903

页数：5

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