Highly diastereoselective hetero-Diels-Alder reactions of alkenyidihydrooxazoles as an approach to novel pyrimidine derivatives

被引：23

作者：

Elliot, MC

Kruiswijk, E

机构：

[1] Department of Chemistry, University of Wales Cardiff, Cardiff CF1 3TB

来源：

CHEMICAL COMMUNICATIONS | 1997年 / 23期

关键词：

D O I：

10.1039/a705571d

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Chiral 2-alkenyldihydrooxazoles react with two equivalents of aryl and arylsulfonyl isocyanates to give chiral non-racemic dihydropyrimidone derivatives in high yield and with complete diastereocontrol.

引用

页码：2311 / 2312

页数：2

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