Total synthesis of nortopsentins A-D, marine alkaloids

被引：0

作者：

Kawasaki, I ^{[1
]}

Yamashita, M ^{[1
]}

Ohta, S ^{[1
]}

机构：

[1] KYOTO PHARMACEUT UNIV, YAMASHIMA KU, KYOTO 607, JAPAN

来源：

CHEMICAL & PHARMACEUTICAL BULLETIN | 1996年 / 44卷 / 10期

关键词：

imidazole; marine alkaloid; Suzuki reaction; palladium catalyst; arylboronic acid; nortopsentin;

D O I：

暂无

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Nortopsentins A-D, antifungal 1,4-bisindolylimidazole marine alkaloids isolated from a sponge, were synthesized through palladium-catalyzed cross-coupling of 3-indolylboronic and 6-bromo-3-indolylboronic acids with halogenoimidazoles as the key reaction.

引用

页码：1831 / 1839

页数：9

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