Facile Syntheses of N-Substituted Imidazoles and Benzotriazoles from Baylis-Hillman Bromides

被引：3
|
作者：
Ye Dongyan [1 ]
Li Jian [1 ]
Li Chunju [1 ]
Jia Xueshun [1 ]
机构：
[1] Shanghai Univ, Dept Chem, Shanghai 200444, Peoples R China
来源：
CHINESE JOURNAL OF CHEMISTRY | 2009年 / 27卷 / 06期
基金：
中国国家自然科学基金;
关键词：
N-substituted imidazole and benzotriazole; Baylis-Hillman bromide; synthesis; EFFICIENT SYNTHESIS; ADDUCTS; ACETATES;
D O I：
10.1002/cjoc.200990194
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A facile synthesis of N-substituted imidazole and benzotriazole derivatives from Baylis-Hillman bromides with imidazole and benzotriazole at room temperature was reported. In view of the simple operation, mild reaction conditions, good to excellent yields, good regio- and stereoselectivity, the present method exhibited its superiority.
引用
收藏
页码：1159 / 1162
页数：4
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