A convenient synthesis of (1S)-tert-butyl-1,2-ethylenediamine

被引：7

作者：

Busacca, CA ^{[1
]}

Grossbach, D ^{[1
]}

Spinelli, E ^{[1
]}

机构：

[1] Boehringer Ingelheim Pharmaceut Inc, Dept Chem Dev, Ridgefield, CT 06877 USA

来源：

TETRAHEDRON-ASYMMETRY | 2000年 / 11卷 / 09期

关键词：

D O I：

10.1016/S0957-4166(00)00145-2

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

A practical four-step synthesis of (1S)-tert-butyl-1,2-ethylenediamine has been developed. The sequence proceeds in good overall yield via crystalline intermediates and provides the title compound in 99.3% ee. (C) 2000 Elsevier Science Ltd. All rights reserved.

引用

页码：1907 / 1910

页数：4

共 20 条

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