Reaction of polychloroacetaldehyde arylsulfonylimines with 2-amino-6H-1,3-thiazine-6-thiones and 2-amino-4-phenyl-6H-1,3-thiazin-6-one

被引：0

作者：

Kaliev, A. R. ^{[1
]}

Serykh, V. Yu ^{[1
]}

Levkovskaya, G. G. ^{[1
]}

Potkin, V. I. ^{[2
]}

Petkevich, S. K. ^{[1
]}

Rozentsveig, I. B. ^{[1
]}

机构：

[1] Russian Acad Sci, Favorskii Irkutsk Inst Chem, Siberian Branch, Ul Favorskogo 1, Irkutsk 664033, Russia

[2] Natl Acad Sci Belarus, Inst Phys Organ Chem, Minsk, BELARUS

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2016年 / 52卷 / 11期

关键词：

N-(2,2-DICHLORO-2-PHENYLETHYLIDENE)ARENESULFONAMIDES; SULFONAMIDES;

D O I：

10.1134/S1070428016110208

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-Amino-4-R-6H-1,3-thiazine-6-thiones and 2-amino-4-phenyl-6H-1,3-thiazin-6-one react with highly electrophilic N-arylsulfonylimines of chloral and phenyldichloroacetic aldehyde at the exocyclic amino group affording in good yields products of nucleophilic addition to the azomethine group of imines: N-[2-polychloro-1-(6-thioxo-4-R-6H-1,3-thiazin-2-ylamino)ethyl]- or -[2-polychloro-1-(6-oxo-4-phenyl-6H-1,3-thiazin-2-ylamino)ethyl]arenesulfonamides.

引用

页码：1670 / 1673

页数：4

共 36 条

[1] N-(2,2,2-trichloroethylidene)- and N-(1-hydroxy-2,2,2-trichloroethyl)amides in C-amidoalkylation reaction of functionally-substituted aromatic compounds
Aizina, YA
Rozentsweig, IB
Levkovskaya, GG
Rozentsweig, GN
Mirskova, AN
[J]. RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2002, 38 (02) : 235 - 238
[2] Synthesis of Binaphthyl Sulfonimides and Their Application in the Enantioselective Michael Addition of Ketones to Nitroalkenes
Ban, Shurong
Du, Da-Ming
Liu, Han
Yang, Wen
[J]. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2010, 2010 (27) : 5160 - 5164
[3] Barton D., 1979, COMPREHENSIVE ORGANI, V3, P5
[4] Barton D., 1979, COMPREHENSIVE ORGANI, V9
[5] Sulfonamides: a patent review (2008-2012)
Carta, Fabrizio
Scozzafava, Andrea
Supuran, Claudiu T.
[J]. EXPERT OPINION ON THERAPEUTIC PATENTS, 2012, 22 (07) : 747 - 758
[6] De Kimpe N., 1988, ALPHA HALOALDEHYDES
[7] REACTIVITY OF ALPHA-HALOGENATED IMINO COMPOUNDS
DEKIMPE, N
VERHE, R
DEBUYCK, L
SCHAMP, N
[J]. ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 1980, 12 (1-2) : 49 - 180
[8] N-Alkylsulfonamides as Useful Carbon Electrophiles
Gu, Yonghong
Tian, Shi-Kai
[J]. SYNLETT, 2013, 24 (10) : 1170 - 1185
[9] Ivin B.A., 2001, 1 MEZHD K KHIM BIOL, V1, P85
[10] Kaluzhskikh A.N., 1997, RUSS J GEN CHEM+, V67, P1126

← 1 2 3 4 →