Synthesis of 2-(aryl methylene)-(1H)-indane-1,3-(2H)-diones as potential fungicidal and bactericidal agents

被引：0

作者：

Meena, S. ^{[1
]}

Shankar, D. ^{[1
]}

Ramseshu, K. V. ^{[1
]}

Giles, D. ^{[1
]}

Prakash, M. S. ^{[1
]}

Venkataraman, S. ^{[1
]}

机构：

[1] KM Coll Pharm, Dept Pharmaceut Chem, Madurai 625107, Tamil Nadu, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2006年 / 45卷 / 06期

关键词：

indanediones; indane-1,3-dione; aldehyde derivatives; synthesis; antifungal activity; antibacterial activity;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction of diethyl phthalate 1 and ethyl acetate 2 in the presence of sodium metal and ethanol affords indane-1, 3-dione 3, which have been substituted at C-2 position with different aromatic aldehydes 4, to yield their respective aryl derivatives of indane-1,3-dione 5a-h. These derivatives are evaluated for their antifungal and antibacterial activity. The structures of all the compounds are determined by IR, H-1 NMR and mass spectrometry.

引用

页码：1572 / 1575

页数：4

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