An Efficient and Stereoselective Synthesis of Pyrazolo[4,3-c]pyridine Derivatives under Microwave Heating

被引：5
作者：
Peng, Ju-Hua [1 ]
Hao, Wen-Juan [1 ]
Tu, Shu-Jiang [1 ]
机构：
[1] Lianyungang Teachers Coll, Lianyungang 222006, Jiangsu, Peoples R China
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2009年 / 46卷 / 05期
基金：
美国国家科学基金会;
关键词：
ASSISTED ORGANIC-SYNTHESIS; MANNICH-TYPE REACTION; ONE-POT; CHEMISTRY; PYRIDINE; DESIGN; WATER;
D O I：
10.1002/jhet.169
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A practical, inexpensive, and rapid method for the stereoselective synthesis of pyrazolo[4,3-c]pyridine derivatives via microwave-assisted reactions of 3,5-diarylidenepiperidin-4-ones with phenylhydrazine in ethylene glycol. This method has the advantages of good yield, operational simplicity, and simple purification procedure.
引用
收藏
页码：849 / 853
页数：5
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