Synthesis of novel 2-azabicyclo[3.1.1]heptane-5-carboxylic acid

被引：1

作者：

He, Shuwen ^{[1
]}

Hao, Jinsong ^{[1
]}

Ashley, Eric R. ^{[1
]}

Chobanian, Harry R. ^{[1
]}

Pio, Barbara ^{[1
]}

Colletti, Steven L. ^{[1
]}

Miller, Michael ^{[1
]}

机构：

[1] Merck Res Labs, Discovery Chem, 2000 Galloping Hill Rd, Kenilworth, NJ 07033 USA

来源：

TETRAHEDRON LETTERS | 2016年 / 57卷 / 11期

关键词：

2-Azabicyclo[3.1.1]heptane-5-carboxylic acid; Amino acid; Bicyclic compound; SUBSTITUTION; DIVERSITY;

D O I：

10.1016/j.tetlet.2016.02.024

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1268 / 1269

页数：2

共 18 条

[1] 2,4-METHANOPROLINE (2-CARBOXY-2,4-METHANOPYRROLIDINE) AND 2,4-METHANOGLUTAMIC ACID (1-AMINO-1,3-DICARBOXYCYCLOBUTANE) IN SEEDS OF ATELEIA-HERBERT-SMITHII PITTIER (LEGUMINOSAE)
BELL, EA
QURESHI, MY
PRYCE, RJ
JANZEN, DH
LEMKE, P
CLARDY, J
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (04) : 1409 - 1412
[2] Synthesis of a Variety of 2-Alkyl-2-Azabicyclo[3.1.1]heptane-1-carbonitriles via a Dynamic Addition-Intramolecular Substitution Sequence
De Blieck, Ann
Stevens, Christian V.
[J]. SYNLETT, 2011, (12) : 1748 - 1752
[3] Elend D., 2005, SYNTHETIC COMMUN, V35, P3151
[4] Stereoselective synthesis of 2,4-methanoproline homologues
Grygorenko, EO
Artamonov, ES
Palamarchuk, GV
Zubatyuk, RI
Shishkin, OV
Komarov, IV
[J]. TETRAHEDRON-ASYMMETRY, 2006, 17 (02) : 252 - 258
[5] TOTAL SYNTHESIS OF CYCLOBUTANE AMINO-ACIDS FROM ATELIA-HERBERT-SMITHII
HUGHES, P
CLARDY, J
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1988, 53 (20) : 4793 - 4796
[6] SYNTHESIS OF 2,4-METHANOPROLINE
HUGHES, P
MARTIN, M
CLARDY, J
[J]. TETRAHEDRON LETTERS, 1980, 21 (48) : 4579 - 4580
[7] Complex-induced proximity effects.: Temperature-dependent regiochemical diversity in lithiation-electrophilic substitution reactions of N-BOC-2-azabicyclo[2.1.1] hexane.: 2,4-and 3,5-methanoprolines
Krow, GR
Herzon, SB
Lin, GL
Qiu, F
Sonnet, PE
[J]. ORGANIC LETTERS, 2002, 4 (18) : 3151 - 3154
[8] A novel synthesis of 2-azabicyclo[2.1.1]hexane from pyridine
Krow, GR
Lee, YB
Lester, WS
Christian, H
Shaw, DA
Yuan, J
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1998, 63 (23) : 8558 - 8560
[9] Park T. H., 1999, PCT Int. Appl., Patent No. [9907706, 18, 9907706]
[10] TOTAL SYNTHESIS OF 2,4-METHANOPROLINE
PIRRUNG, MC
[J]. TETRAHEDRON LETTERS, 1980, 21 (48) : 4577 - 4578

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