共 6 条
[1]
Safety and efficacy of the HIV-1 integrase inhibitor raltegravir (MK-0518) in treatment-experienced patients with multidrug-resistant virus: a phase II randomised controlled trial
[J].
Grinsztejn, Beatriz
;
Nguyen, Bach-Yen
;
Katlama, Christine
;
Gatell, Jose M.
;
Lazzarin, Adriano
;
Vittecoq, Daniel
;
Gonzalez, Charles J.
;
Chen, Joshua
;
Harvey, Charlotte M.
;
Isaacs, Robin D.
.
LANCET,
2007, 369 (9569)
:1261-1269

Grinsztejn, Beatriz
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Nguyen, Bach-Yen
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Katlama, Christine
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Gatell, Jose M.
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Lazzarin, Adriano
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Vittecoq, Daniel
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Gonzalez, Charles J.
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Chen, Joshua
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Harvey, Charlotte M.
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil

Isaacs, Robin D.
论文数: 0 引用数: 0
h-index: 0
机构: Fundacao Oswaldo Cruz, Evandro Chagas Clin Res Inst, Rio De Janeiro, Brazil
[2]
Safety, tolerability, and pharmacokinetics of raltegravir after single and multiple doses in healthy subjects
[J].
Iwamoto, M.
;
Wenning, L. A.
;
Petry, A. S.
;
Laethem, M.
;
De Smet, M.
;
Kost, J. T.
;
Merschman, S. A.
;
Strohmaier, K. M.
;
Ramael, S.
;
Lasseter, K. C.
;
Stone, J. A.
;
Gottesdiener, K. M.
;
Wagner, J. A.
.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
2008, 83 (02)
:293-299

Iwamoto, M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Wenning, L. A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Petry, A. S.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Laethem, M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

De Smet, M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Kost, J. T.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Merschman, S. A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Strohmaier, K. M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Ramael, S.
论文数: 0 引用数: 0
h-index: 0
机构:
SGS Life Sci Serv, Antwerp, Belgium Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Lasseter, K. C.
论文数: 0 引用数: 0
h-index: 0
机构:
Pharmaceut Dev Grp, Miami, FL USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Stone, J. A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Gottesdiener, K. M.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA

Wagner, J. A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
Div Merck & Co Inc, Merck Res Labs, Dept Clin Drug Metab, White House Stn, NJ USA
Div Merck & Co Inc, Merck Res Labs, Dept Med Commun, White House Stn, NJ USA Merck Res Labs, Dept Clin Pharmacol, Div Merck & Co Inc, White House Stn, NJ 08889 USA
[3]
Safety and efficacy of raltegravir-based versus efavirenz-based combination therapy in treatment-naive patients with HIV-1 infection: a multicentre, double-blind randomised controlled trial
[J].
Lennox, Jeffrey L.
;
Dejesus, Edwin
;
Lazzarin, Adriano
;
Pollard, Richard B.
;
Ramalho Madruga, Jose Valdez
;
Berger, Daniel S.
;
Zhao, Jing
;
Xu, Xio
;
Williams-Diaz, Angela
;
Rodgers, Anthony J.
;
Barnard, Richard J. O.
;
Miller, Michael D.
;
DiNubile, Mark J.
;
Nguyen, Bach-Yen
;
Leavitt, Randi
;
Sklar, Peter
.
LANCET,
2009, 374 (9692)
:796-806

Lennox, Jeffrey L.
论文数: 0 引用数: 0
h-index: 0
机构:
Emory Univ, Sch Med, Atlanta, GA USA Merck Res Labs, N Wales, PA 19454 USA

Dejesus, Edwin
论文数: 0 引用数: 0
h-index: 0
机构:
Orlando Immunol Ctr, Orlando, FL USA Merck Res Labs, N Wales, PA 19454 USA

Lazzarin, Adriano
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Vita Salute San Raffaele, Milan, Italy Merck Res Labs, N Wales, PA 19454 USA

Pollard, Richard B.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Davis, Sacramento, CA 95817 USA Merck Res Labs, N Wales, PA 19454 USA

Ramalho Madruga, Jose Valdez
论文数: 0 引用数: 0
h-index: 0
机构:
Ctr Referencia & Treinamento DST AIDS, Sao Paulo, Brazil Merck Res Labs, N Wales, PA 19454 USA

Berger, Daniel S.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Illinois, Northstar Med Ctr, Chicago, IL USA Merck Res Labs, N Wales, PA 19454 USA

Zhao, Jing
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Xu, Xio
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Williams-Diaz, Angela
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Rodgers, Anthony J.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Barnard, Richard J. O.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Miller, Michael D.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

DiNubile, Mark J.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Nguyen, Bach-Yen
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Leavitt, Randi
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA

Sklar, Peter
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, N Wales, PA 19454 USA Merck Res Labs, N Wales, PA 19454 USA
[4]
Rapid and durable Antiretroviral effect of the HIV-1 integrase inhibitor raltegravir as part of combination therapy in treatment-naive patients with HIV-1 infection - Results of a 48-week controlled study
[J].
Markowitz, Martin
;
Nguyen, Bach-Yen
;
Gotuzzo, Eduardo
;
Mendo, Fernando
;
Ratanasuwan, Winai
;
Kovacs, Colin
;
Prada, Guillermo
;
Morales-Ramirez, Javier O.
;
Crumpacker, Clyde S.
;
Isaacs, Robin D.
;
Gilde, Lucinda R.
;
Wan, Hong
;
Miller, Michael D.
;
Wenning, Larissa A.
;
Teppler, Hedy
.
JAIDS-JOURNAL OF ACQUIRED IMMUNE DEFICIENCY SYNDROMES,
2007, 46 (02)
:125-133

Markowitz, Martin
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Nguyen, Bach-Yen
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Gotuzzo, Eduardo
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Mendo, Fernando
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Ratanasuwan, Winai
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Kovacs, Colin
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Prada, Guillermo
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Morales-Ramirez, Javier O.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Crumpacker, Clyde S.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Isaacs, Robin D.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Gilde, Lucinda R.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Wan, Hong
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Miller, Michael D.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Wenning, Larissa A.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA

Teppler, Hedy
论文数: 0 引用数: 0
h-index: 0
机构: Merck Res Labs, N Wales, PA 19454 USA
[5]
Antiretroviral activity, pharmacokinetics, and tolerability of MK-0518, a novel inhibitor of HIV-1 integrase, dosed as monotherapy for 10 days in treatment-naive HIV-1-infected individuals
[J].
Markowitz, Martin
;
Morales-Ramirez, Javier O.
;
Nguyen, Bach-Yen
;
Kovacs, Colin M.
;
Steigbigel, Roy T.
;
Cooper, David A.
;
Liporace, Ralph
;
Schwartz, Robert
;
Isaacs, Robin
;
Gilde, Lucinda R.
;
Penning, Larissa
;
Zhao, Jing
;
Teppler, Hedy
.
JAIDS-JOURNAL OF ACQUIRED IMMUNE DEFICIENCY SYNDROMES,
2006, 43 (05)
:509-515

Markowitz, Martin
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Morales-Ramirez, Javier O.
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Nguyen, Bach-Yen
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Kovacs, Colin M.
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Steigbigel, Roy T.
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Cooper, David A.
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Liporace, Ralph
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Schwartz, Robert
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Isaacs, Robin
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Gilde, Lucinda R.
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Penning, Larissa
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Zhao, Jing
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA

Teppler, Hedy
论文数: 0 引用数: 0
h-index: 0
机构: Rockefeller Univ, Aaron Diamond AIDS Res Ctr, New York, NY 10021 USA
[6]
NEELY M, 2009, 5 IAS C HIV PATH CAP