SAFETY AND EFFICACY OF ABT-494, A NOVEL SELECTIVE JAK1 INHIBITOR, IN PATIENTS WITH ACTIVE RHEUMATOID ARTHRITIS WITH AN INADEQUATE RESPONSE TO METHOTREXATE

被引:1
|
作者
Genovese, M. C. [1 ]
Smolen, J. S. [2 ,3 ]
Weinblatt, M. E. [4 ]
Meerwein, S. [5 ]
Camp, H. S. [5 ]
Wang, L. [5 ]
Othman, A. A. [5 ]
Khan, N. [5 ]
Jungerwirth, S. [5 ]
机构
[1] Stanford Univ, Sch Med, Palo Alto, CA 94304 USA
[2] Med Univ Vienna, Vienna, Austria
[3] Hietzing Hosp, Vienna, Austria
[4] Brigham & Womens Hosp, 75 Francis St, Boston, MA 02115 USA
[5] AbbVie Inc, N Chicago, IL USA
关键词
D O I
10.1136/annrheumdis-2016-eular.3698
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
OP0223
引用
收藏
页码:141 / 142
页数:2
相关论文
共 50 条
  • [1] Efficacy and Safety of ABT-494, a Selective JAK-1 Inhibitor, in a Phase IIb Study in Patients With Rheumatoid Arthritis and an Inadequate Response to Methotrexate
    Genovese, Mark C.
    Smolen, Josef S.
    Weinblatt, Michael E.
    Burmester, Gerd R.
    Meerwein, Sebastian
    Camp, Heidi S.
    Wang, Li
    Othman, Ahmed A.
    Khan, Nasser
    Pangan, Aileen L.
    Jungerwirth, Steven
    ARTHRITIS & RHEUMATOLOGY, 2016, 68 (12) : 2857 - 2866
  • [2] SAFETY AND EFFICACY OF ABT-494, A NOVEL SELECTIVE JAK1 INHIBITOR, IN PATIENTS WITH ACTIVE RHEUMATOID ARTHRITIS AND INADEQUATE RESPONSE OR INTOLERANCE TO ANTI-TNF BIOLOGIC THERAPY
    Kremer, J. M.
    Keystone, E. C.
    Emery, P.
    Camp, H. S.
    Friedman, A.
    Wang, L.
    Othman, A. A.
    Khan, N.
    Jungerwirth, S.
    ANNALS OF THE RHEUMATIC DISEASES, 2016, 75 : 1038 - 1039
  • [3] Safety and Efficacy of ABT-494, a Novel Selective JAK1 Inhibitor, in Patients with Active Rheumatoid Arthritis and Inadequate Response or Intolerance to Anti-TNF Biologic Therapy
    Kremer, Joel M.
    Keystone, Edward C.
    Emery, Paul
    Camp, Heidi S.
    Friedman, Alan
    Wang, Li
    Othman, Ahmed A.
    Khan, Nasser
    Jungerwirth, Steven
    ARTHRITIS & RHEUMATOLOGY, 2015, 67
  • [4] PHARMACOKINETICS, SAFETY AND TOLERABILITY OF THE SELECTIVE JAK1 INHIBITOR, ABT-494, IN HEALTHY VOLUNTEERS AND SUBJECTS WITH RHEUMATOID ARTHRITIS
    Mohamed, M. -E.
    Camp, H.
    Jiang, P.
    Padley, R.
    Asatryan, A.
    Othman, A. A.
    ANNALS OF THE RHEUMATIC DISEASES, 2015, 74 : 258 - 258
  • [5] Pharmacokinetics, Safety and Tolerability of ABT-494, a Novel Selective JAK 1 Inhibitor, in Healthy Volunteers and Subjects with Rheumatoid Arthritis
    Mohamed, Mohamed-Eslam F.
    Camp, Heidi S.
    Jiang, Ping
    Padley, Robert J.
    Asatryan, Armen
    Othman, Ahmed A.
    CLINICAL PHARMACOKINETICS, 2016, 55 (12) : 1547 - 1558
  • [6] Pharmacokinetics, Safety and Tolerability of ABT-494, a Novel Selective JAK 1 Inhibitor, in Healthy Volunteers and Subjects with Rheumatoid Arthritis
    Mohamed-Eslam F. Mohamed
    Heidi S. Camp
    Ping Jiang
    Robert J. Padley
    Armen Asatryan
    Ahmed A. Othman
    Clinical Pharmacokinetics, 2016, 55 : 1547 - 1558
  • [7] Characterization of ABT-494, a Second Generation Jak1 Selective Inhibitor.
    Graff, Candace
    Schwartz, Annette
    Voss, Jeffrey
    Wishart, Neil
    Olson, Lisa
    George, Jonathon
    Hyland, Deborah
    Camp, Heidi
    ARTHRITIS & RHEUMATOLOGY, 2014, 66 : S659 - S660
  • [8] A Phase IIb Study of ABT-494, a Selective JAK-1 Inhibitor, in Patients With Rheumatoid Arthritis and an Inadequate Response to Anti-Tumor Necrosis Factor Therapy
    Kremer, Joel M.
    Emery, Paul
    Camp, Heidi S.
    Friedman, Alan
    Wang, Li
    Othman, Ahmed A.
    Khan, Nasser
    Pangan, Aileen L.
    Jungerwirth, Steven
    Keystone, Edward C.
    ARTHRITIS & RHEUMATOLOGY, 2016, 68 (12) : 2867 - 2877
  • [9] SAFETY AND EFFICACY OF ABT-494 (UPADACITINIB), AN ORAL JAK1 INHIBITOR, AS INDUCTION THERAPY IN PATIENTS WITH CROHN'S DISEASE: RESULTS FROM CELEST
    Sandborn, William J.
    Feagan, Brian G.
    Panes, Julian
    D'Haens, Geert R.
    Colombel, Jean Frederic
    Zhou, Qian
    Huang, Bidan
    Enejosa, Jeffrey V.
    Pangan, Aileen L.
    Lacerda, Ana P.
    GASTROENTEROLOGY, 2017, 152 (05) : S1308 - S1309
  • [10] Long-Term Safety and Efficacy of Upadacitinib (ABT-494), an Oral JAK-1 Inhibitor in Patients with Rheumatoid Arthritis in an Open Label Extension Study
    Genovese, Mark C.
    Kremer, Joel
    Zhong, Sheng
    Friedman, Alan
    ARTHRITIS & RHEUMATOLOGY, 2017, 69