Synthesis and evaluation of novel 1H-pyrrolo[2,3-b] pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3 (vol 23, pg 4871, 2015)

被引:0
作者
Nakajima, Yutaka [1 ]
Inoue, Takayuki [1 ]
Nakai, Kazuo [1 ]
Mukoyoshi, Koichiro [1 ]
Hamaguchi, Hisao [1 ]
Hatanaka, Keiko [1 ]
Sasaki, Hiroshi [1 ]
Tanaka, Akira [1 ]
Takahashi, Fumie [1 ]
Kunikawa, Shigeki [1 ]
Usuda, Hiroyuki [1 ]
Moritomo, Ayako [1 ]
Higashi, Yasuyuki [1 ]
Inami, Masamichi [1 ]
Shirakami, Shohei [1 ]
机构
[1] Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan
关键词
D O I
10.1016/j.bmc.2017.03.043
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:2813 / 2813
页数:1
相关论文
共 1 条
  • [1] Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3
    Nakajima, Yutaka
    Inoue, Takayuki
    Nakai, Kazuo
    Mukoyoshi, Koichiro
    Hamaguchi, Hisao
    Hatanaka, Keiko
    Sasaki, Hiroshi
    Tanaka, Akira
    Takahashi, Fumie
    Kunikawa, Shigeki
    Usuda, Hiroyuki
    Moritomo, Ayako
    Higashi, Yasuyuki
    Inami, Masamichi
    Shirakami, Shohei
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (15) : 4871 - 4883