Cyanoacetanilides Intermediates in Heterocyclic Synthesis. Part 5: Preparation of Hitherto Unknown 5-Aminopyrazole and Pyrazolo[1,5-a]pyrimidine Derivatives Containing Sulfamoyl Moiety

被引:28
作者
Ammar, Yousry A. [2 ]
Aly, Mohsen M. [2 ]
Al-Sehemi, Abd Allah G. [3 ]
Salem, Mohamed A. [2 ]
El-Gaby, Mohamed S. A. [1 ]
机构
[1] Al Azhar Univ, Dept Chem, Fac Sci, Assiut 71524, Egypt
[2] Al Azhar Univ, Dept Chem, Fac Sci, Nasr City, Cairo, Egypt
[3] Teachers Coll, Dept Chem, Abha, Saudi Arabia
关键词
5-Aminopyrazole; Pyrazolo[1,5-a]pyrimidines; Sulfonamides; Cyanoacetamide; ACTIVATED NITRILES; FACILE SYNTHESIS;
D O I
10.1002/jccs.200900154
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Novel 5-aminopyrazole and pyrazolo[1,5-a]pyrimidine derivatives have been synthesized from the readily accessible cyanoacetanilide derivative (2).
引用
收藏
页码:1064 / 1071
页数:8
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