Synthesis of biologically active benzothiazole substituted thiazolidinone derivatives via cyclization of unsymmetrical imines

被引：0

作者：

Nagarajan, Arasampattu S. ^{[1
]}

Kamalraj, S. ^{[2
]}

Muthumary, J. ^{[2
]}

Reddy, Boreddy S. R. ^{[1
]}

机构：

[1] Cent Leather Res Inst, Ind Chem Lab, Madras 600020, Tamil Nadu, India

[2] Univ Madras, Ctr Adv Studies Bot, Madras 600025, Tamil Nadu, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2009年 / 48卷 / 11期

关键词：

Unsymmetrical imine; benzothiazole; thiazolidinone; cyclization; antibacterial activity; ANTIMICROBIAL ACTIVITY; AGENTS; 4-THIAZOLIDINONES;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Novel benzothiazole substituted thiazolidinone derivatives are synthesized through cyclisation of unsymmetrical imine with mercaptoacid in the presence of SnCl2 center dot 2H(2)O and evaluated their inhibition ability against Proteus mirabilis, Staphylococcus aureus, Salmonella typhi and Klebsiella pneumoniae.

引用

页码：1577 / 1582

页数：6

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