Synthesis and acaricidal activities of new 2-polyfluorophenylbenzazole derivatives

被引:0
作者
Mouri, T
Tokumura, J
Kochi, S
Fukui, H
Nakano, J
Ando, T
Hori, M
机构
[1] Kaken Pharmaceut Co Ltd, Fujieda, Shizuoka 4268646, Japan
[2] Kaken Pharmaceut Co Ltd, Bunkyo Ku, Tokyo 1138650, Japan
[3] Kaken Pharmaceut Co Ltd, Yamashina Ku, Kyoto 6078042, Japan
[4] Tokyo Univ Agr & Technol, Grad Sch Bioapplicat & Syst Engn, Koganei, Tokyo 1848588, Japan
来源
JOURNAL OF PESTICIDE SCIENCE | 2002年 / 27卷 / 04期
关键词
benzoxazole; benzothiazole; acaricidal activity; two-spotted spider mite; ovicide;
D O I
暂无
中图分类号
Q96 [昆虫学];
学科分类号
摘要
New 2-phenylbenzazole derivatives, thirteen benzoxazoles and eight benzothiazoles, were synthesized, and their acaricidal activities measured against the two-spotted spider mite (TSM). Some compounds with a polyfluorophenyl group were highly effective in killing the eggs (LC50: < 50 ppm) with moderate activity (LC50: 150-200 ppm) against the adults. Among them, 2-(3-chloro-2,4,5-trifluorophenyl)-5-methylbenzoxazole was selected as the most promising candidate for an acaricide, and the effects of its concentrate were evaluated. This formulation achieved a high rate of mortality in the citrus red mite and a kelthane-resistant strain of TSM in addition to a common strain of TSM.
引用
收藏
页码:353 / 359
页数:7
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