SYNTHESIS OF NEW 3-CARBOXAMIDINE IMINOCOUMARINS AND BENZOPYRANO[2,3-d]PYRIMIDINES

被引：0

作者：

Trichili, Sihem ^{[1
]}

Kammoun, Myriam ^{[1
]}

Turki-Guermazi, Hamida ^{[1
]}

Abid, Souhir ^{[1
]}

Ammar, Houcine ^{[1
]}

机构：

[1] Univ Sfax, Fac Sci Sfax, Lab Chim Appl Heterocycles Corps Gras & Polymeres, Sfax 3000, Tunisia

来源：

SYNTHETIC COMMUNICATIONS | 2015年 / 45卷 / 08期

关键词：

Anticholinesterase activity; benzopyrano[2,3-d]pyrimidines; carboxamidines; iminocoumarins; FLUORESCENT IMINOCOUMARINS; PHARMACOLOGICAL EVALUATION; OPTICAL-PROPERTIES; ANTIPLATELET; SERIES; DERIVATIVES;

D O I：

10.1080/00397911.2014.997365

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new approach to synthesis of a series of 3-carboxamidine iminocoumarins derivatives and substituted benzopyrano[2,3-d]pyrimidines was developed. The chemical structure of all the compounds was investigated by infrared, H-1 NMR, C-13 NMR, mass, and elemental analysis. The anticholinesterase activity of compound 12 was evaluated according to the modified Ellman's method.

引用

页码：958 / 966

页数：9

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