An asymmetric aminohydroxylation route to (+)-L-733,060

被引：21

作者：

Kandula, SRV ^{[1
]}

Kumar, P ^{[1
]}

机构：

[1] Natl Chem Lab, Div Organ Chem, Pune 411008, Maharashtra, India

来源：

TETRAHEDRON-ASYMMETRY | 2005年 / 16卷 / 21期

关键词：

D O I：

10.1016/j.tetasy.2005.09.010

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

An enantioselective synthesis of (+)-L-733,060 starting from cinnamic acid using Sharpless asymmetric aminohydroxylation and Wittig reactions as the key steps is described. (c) 2005 Elsevier Ltd. All rights reserved.

引用

页码：3579 / 3583

页数：5

共 39 条

[1]

Baker R., 1993, Eur. Patent, Patent No. [528495, 0528495A1, 0528495]

[2] Stereoselective synthesis of L-733,060 [J].

Bhaskar, G ;

Rao, BV .

TETRAHEDRON LETTERS, 2003, 44 (05) :915-917

[3]

Bodas Mandar S., 2004, TETRAHEDRON LETT, V45, P987

[4] An asymmetric dihydroxylation route to (2S,3S)-3-hydroxypipecolic acid [J].

Bodas, MS ;

Kumar, P .

TETRAHEDRON LETTERS, 2004, 45 (46) :8461-8463

[5] N-bromoacetamide - A new nitrogen source for the catalytic asymmetric aminohydroxylation of olefins [J].

Bruncko, M ;

Schlingloff, G ;

Sharpless, KB .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1997, 36 (13-14) :1483-1486

[6] Stereoselective synthesis of (2S,3S)-3-hydroxy-2-phenylpiperidines, precursors of non-peptidic substance P antagonists [J].

Calvez, O ;

Langlois, N .

TETRAHEDRON LETTERS, 1999, 40 (39) :7099-7100

[7]

Fernandes RA, 2003, SYNTHESIS-STUTTGART, P129

[8]

Fernandes RA, 2002, EUR J ORG CHEM, V2002, P2921, DOI 10.1002/1099-0690(200209)2002:17<2921::AID-EJOC2921>3.0.CO

[9]

2-N

[10]

Fernandes RA, 2000, EUR J ORG CHEM, V2000, P3447

← 1 2 3 4 →