Facile one-pot synthesis of aromatic and heteroaromatic sulfonamides

被引：119

作者：

Pandya, R ^{[1
]}

Murashima, T ^{[1
]}

Tedeschi, L ^{[1
]}

Barrett, AGM ^{[1
]}

机构：

[1] Univ London Imperial Coll Sci Technol & Med, Dept Chem, London SW7 2AZ, England

来源：

JOURNAL OF ORGANIC CHEMISTRY | 2003年 / 68卷 / 21期

关键词：

D O I：

10.1021/jo034643j

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of arene and heteroarene sulfonamides were prepared in one vessel from aryl and heteroaryl bromides via conversion into the corresponding Grignard reagents using either magnesium or isopropylmagnesium chloride and subsequent reaction with sulfur dioxide, sulfuryl chloride, and an amine.

引用

页码：8274 / 8276

页数：3

共 18 条

[1] Preparation of new polyfunctional magnesiated heterocycles using a chlorine-, bromine-, or iodine-magnesium exchange [J].

Abarbri, M ;

Thibonnet, J ;

Bérillon, L ;

Dehmel, F ;

Rottländer, M ;

Knochel, P .

JOURNAL OF ORGANIC CHEMISTRY, 2000, 65 (15) :4618-4634

[2]

Abarbri M, 1999, SYNLETT, P1577

[3]

Anderson KK, 1979, SULFONIC ACIDS THEIR, V3, P331

[4]

Bérillon L, 1998, SYNLETT, P1359

[5] PREPARATION OF ARENESULPHONYL CHLORIDES FROM GRIGNARD REAGENTS [J].

BHATTACHARYA, SN ;

EABORN, C ;

WALTON, DRM .

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1968, (10) :1265-+

[6]

Boudier A, 2000, ANGEW CHEM INT EDIT, V39, P4414, DOI 10.1002/1521-3773(20001215)39:24<4414::AID-ANIE4414>3.0.CO

[7]

2-C

[8]

Boymond L, 1998, ANGEW CHEM INT EDIT, V37, P1701, DOI 10.1002/(SICI)1521-3773(19980703)37:12<1701::AID-ANIE1701>3.0.CO

[9]

2-U

[10]

CREMLYN R, 1996, ORGANOSULFUR CHEM IN, P224

← 1 2 →