A versatile one-pot synthesis of 4-aryl-1,5-disubstituted 1,2,3-triazoles via 1,3-dipolar cycloaddition followed by Negishi reaction under new conditions

被引：24
作者：
Akao, Atsushi
Tsuritani, Takayuki
Kii, Satoshi
Sato, Kimihiko
Nonoyama, Nobuaki
Mase, Toshiaki
Yasuda, Nobuyoshi
机构：
[1] Merck Res Labs, Tsukuba, Ibaraki 3002611, Japan
[2] Merck Res Labs, Dept Proc Res, Rahway, NJ 07065 USA
来源：
SYNLETT | 2007年 / 01期
关键词：
triazole; Negishi reaction; 1,3-dipolar cycloaddition; XANTPHOS; zinc; cross-coupling;
D O I：
10.1055/s-2006-958435
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Several derivatives of 4-aryl-1,5-disubstituted 1,2,3-triazole were synthesized in good yields via 1,3-dipolar cycloaddition followed by Negishi reaction under new conditions.
引用
收藏
页码：31 / 36
页数：6
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