SYNTHESIS OF NITROGEN-CONTAINING HETEROCYCLES USING CONJUGATE ADDITION REACTIONS OF NUCLEOPHILES TO α,β-UNSATURATED IMINES

被引：10

作者：

Hachiya, Iwao ^{[1
]}

Mizota, Isao ^{[1
]}

Shimizu, Makoto ^{[1
]}

机构：

[1] Mie Univ, Grad Sch Engn, Dept Chem Mat, Tsu, Mie 5148507, Japan

来源：

HETEROCYCLES | 2012年 / 85卷 / 05期

基金：

日本科学技术振兴机构;

关键词：

2,3,5-Trisubstituted Pyrrole; delta-Lactam; 2-Pyridone; 2-Iminopyridine; beta-Lactam; KETENE SILYL (THIO)ACETALS; ANODIC AMIDE OXIDATIONS; FORMAL TOTAL-SYNTHESIS; STEREOSELECTIVE-SYNTHESIS; EFFICIENT SYNTHESIS; RING-EXPANSION; ALKYNYL IMINES; REGIOSELECTIVE SYNTHESIS; SUBSTITUTED PYRROLES; 2-PYRIDONE SYNTHESIS;

D O I：

10.3987/REV-12-726

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthetic methods for the synthesis of nitrogen-containing heterocycles are of utmost interest and importance because these structures are the key components of natural and unnatural biologically active compounds and functionalized materials. This review summarizes the synthesis of nitrogen-containing heterocycles, where the conjugate addition of nucleophiles to alpha,beta-unsaturated i mines is the crucial step.

引用

页码：993 / 1016

页数：24

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