Synthesis of 1,2-dihydropyrrolo[1,2-c]pyrimidin-1-ones

被引：19

作者：

Alvarez, M

Fernández, D

Joule, JA ^{[1
]}

机构：

[1] Univ Barcelona, Fac Farm, Lab Quim Organ, E-08028 Barcelona, Spain

[2] Univ Manchester, Dept Chem, Manchester M13 9PL, Lancs, England

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1999年 / 03期

关键词：

D O I：

10.1039/a809280j

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1,2-Dihydropyrrolo[1,2-c]pyrimidin-1-ones 2 have been synthesised from pyrrole. We have developed a versatile procedure for the introduction of substituents into the pyrrolopyrimidinones 2, at positions 5 or 7 as desired, and as required by our plans-for the synthesis of the variolin type sea alkaloids.

引用

页码：249 / 255

页数：7

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