Protection afforded by methanol extract of Calotropis procera latex in experimental model of colitis is mediated through inhibition of oxidative stress and pro-inflammatory signaling
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作者:
Kumar, Vijay L.
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All India Inst Med Sci, Dept Pharmacol, New Delhi 110029, IndiaAll India Inst Med Sci, Dept Pharmacol, New Delhi 110029, India
Kumar, Vijay L.
[1
]
Pandey, Abhimanu
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All India Inst Med Sci, Dept Pharmacol, New Delhi 110029, IndiaAll India Inst Med Sci, Dept Pharmacol, New Delhi 110029, India
Pandey, Abhimanu
[1
]
Verma, Sneh
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All India Inst Med Sci, Dept Pharmacol, New Delhi 110029, IndiaAll India Inst Med Sci, Dept Pharmacol, New Delhi 110029, India
Verma, Sneh
[1
]
Das, Prasenjit
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All India Inst Med Sci, Dept Pathol, New Delhi 110029, IndiaAll India Inst Med Sci, Dept Pharmacol, New Delhi 110029, India
Das, Prasenjit
[2
]
机构:
[1] All India Inst Med Sci, Dept Pharmacol, New Delhi 110029, India
[2] All India Inst Med Sci, Dept Pathol, New Delhi 110029, India
Calotropis procera, a latex producing plant is known to possess medicinal properties including its beneficial effect in gastrointestinal disorders. The anti-inflammatory effect of its latex in various experimental models is noteworthy and in light of this the present study was carried out with an objective to evaluate its efficacy in ulcerative colitis, an inflammatory condition of the colon. Colitis was induced in rats by acetic acid and the rats were divided into four groups where one group served as experimental control and the other groups were treated with two doses of methanol extract of dried latex of C. procera (MeDL; 50 and 150 mg/kg) and mesalazine (MSZ; 300 mg/kg). The study also included normal control (NC) group for comparison of various parameters related to colon like macroscopic changes, ulcer score, adherent mucus content, weight/length ratio, small intestinal transit, oxidative stress and inflammatory markers, tissue histology and immunoreactivity of cyclooxygenase-2 (COX-2), inducible nitric oxide synthase (iNOS) and nuclear factor kappa beta (NF kappa B) subunit p65. Treatment of colitic rats with MeDL produced a significant reduction in colonic mucosal damage as revealed by macroscopic and microscopic evaluation and normalization of tissue levels of oxidative stress markers and pro-inflammatory mediators. The protection afforded by MeDL was also evident from its restorative effect on tissue histology and expression of COX-2, iNOS and NF kappa B(p65). This study shows that by targeting oxidative stress and NF kappa B(p65) mediated pro-inflammatory signaling, the latex of C. procera affords protection in colitis and its effect was comparable to that of mesalazine. This study suggests that latex of C. procera could serve as a promising therapeutic option for treating inflammatory conditions of the colon.
机构:
Islamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Asadi, Amirhooman
Nezhad, Davood Yaghobi
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Payame Noor Univ, Fac Agr, Dept Agr Biotechnol, Tehran, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Nezhad, Davood Yaghobi
Javazm, Amirreza Rafiei
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Shahid Sadoughi Univ Med Sci, Fac Nursing & Midwifery, Student Res Comm, Yazd, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Javazm, Amirreza Rafiei
Khanicheragh, Parisa
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Lorestan Univ Med Sci, Dept Clin Biochem, Khorramabad, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Khanicheragh, Parisa
Mashouri, Ladan
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Shahrekord Univ, Fac Sci, Dept Genet, Shahrekord, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Mashouri, Ladan
Shakeri, Fatemeh
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Jahrom Univ Med Sci, Jahrom, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Shakeri, Fatemeh
Abbasi, Mojtaba
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Islamic Azad Univ, Fac Vet Med, Shahrekord Branch, Vet Med, Shahrekord, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Abbasi, Mojtaba
Afrazian, Mahya Sadat
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Shiraz Univ, Fac Basic Sci, Dept Biol, Shiraz, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Afrazian, Mahya Sadat
Niknam, Zahra
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Ahvaz Jundishapor Univ Med Sci, Fac Med, Dept Clin Biochem, Student Res Comm, Ahvaz, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
机构:
Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Lim, Jae Sung
Li, Xiangying
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Li, Xiangying
Lee, Da Young
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CUOME BIO Co Ltd, R&D Ctr, Sandan gil, Sandan-gil,Hwasun-eup, Hwasun 58141, Jeonranam Do, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Lee, Da Young
Yao, Lulu
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Yao, Lulu
Yoo, Guijae
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Korea Food Res Inst, 245,Nongsaengmyeong-ro,Iseo-myeon, Wanju 55365, Jeonrabug Do, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Yoo, Guijae
Kim, Yunyeong
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Kim, Yunyeong
Eum, Sang Mi
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Korea Res Inst Biosci & Biotechnol, Int Biol Mat Res Ctr, 125 Gwahak-ro, Daejeon 34141, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Eum, Sang Mi
Cho, Young-Chang
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Cho, Young-Chang
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Yoon, Somy
Park, Su-Jin
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Korea Res Inst Biosci & Biotechnol, Funct Biomat Res Ctr, 181 Ipsin-gil, Jeongeup Si 56212, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
机构:
Natl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Taichung Vet Gen Hosp, Dept Phys Med & Rehabil, Taichung, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Cheng, Yuan-Yang
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Kao, Chung-Lan
Ma, Hsin-I
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Triserv Gen Hosp, Natl Def Med Ctr, Dept Neurol Surg, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Ma, Hsin-I
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Hung, Ching-Hsia
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Wang, Chin-Tien
Liu, Ding-Hao
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Natl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Taipei Vet Gen Hosp, Dept Phys Med & Rehabil, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Liu, Ding-Hao
Chen, Po-Yin
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Taipei Vet Gen Hosp, Dept Phys Med & Rehabil, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Wang, Ning
Yu, Hai
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Yu, Hai
Song, Qian
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Song, Qian
Mao, Ping
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Mao, Ping
Li, Kuo
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Li, Kuo
Bao, Gang
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
机构:
Olabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Alabi, Akinyinka O.
Ajayi, Abayomi M.
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Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Ajayi, Abayomi M.
Ben-Azu, Benneth
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Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, Nigeria
PAMO Univ Med Sci, Fac Basic Med Sci, Dept Pharmacol, Port Harcourt, Rivers State, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Ben-Azu, Benneth
Bakre, Adewale G.
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Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Bakre, Adewale G.
Umukoro, Solomon
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Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
机构:
Islamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Asadi, Amirhooman
Nezhad, Davood Yaghobi
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h-index: 0
机构:
Payame Noor Univ, Fac Agr, Dept Agr Biotechnol, Tehran, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Nezhad, Davood Yaghobi
Javazm, Amirreza Rafiei
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h-index: 0
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Shahid Sadoughi Univ Med Sci, Fac Nursing & Midwifery, Student Res Comm, Yazd, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Javazm, Amirreza Rafiei
Khanicheragh, Parisa
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h-index: 0
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Lorestan Univ Med Sci, Dept Clin Biochem, Khorramabad, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Khanicheragh, Parisa
Mashouri, Ladan
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Shahrekord Univ, Fac Sci, Dept Genet, Shahrekord, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Mashouri, Ladan
Shakeri, Fatemeh
论文数: 0引用数: 0
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机构:
Jahrom Univ Med Sci, Jahrom, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Shakeri, Fatemeh
Abbasi, Mojtaba
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Islamic Azad Univ, Fac Vet Med, Shahrekord Branch, Vet Med, Shahrekord, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Abbasi, Mojtaba
Afrazian, Mahya Sadat
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h-index: 0
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Shiraz Univ, Fac Basic Sci, Dept Biol, Shiraz, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
Afrazian, Mahya Sadat
Niknam, Zahra
论文数: 0引用数: 0
h-index: 0
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Ahvaz Jundishapor Univ Med Sci, Fac Med, Dept Clin Biochem, Student Res Comm, Ahvaz, IranIslamic Azad Univ, Fac Vet Med, Karaj Branch, Vet Med, Karaj, Iran
机构:
Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Lim, Jae Sung
Li, Xiangying
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h-index: 0
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Li, Xiangying
Lee, Da Young
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h-index: 0
机构:
CUOME BIO Co Ltd, R&D Ctr, Sandan gil, Sandan-gil,Hwasun-eup, Hwasun 58141, Jeonranam Do, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Lee, Da Young
Yao, Lulu
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h-index: 0
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Yao, Lulu
Yoo, Guijae
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h-index: 0
机构:
Korea Food Res Inst, 245,Nongsaengmyeong-ro,Iseo-myeon, Wanju 55365, Jeonrabug Do, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Yoo, Guijae
Kim, Yunyeong
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h-index: 0
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Kim, Yunyeong
Eum, Sang Mi
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h-index: 0
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Korea Res Inst Biosci & Biotechnol, Int Biol Mat Res Ctr, 125 Gwahak-ro, Daejeon 34141, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Eum, Sang Mi
Cho, Young-Chang
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h-index: 0
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Chonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
Cho, Young-Chang
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Yoon, Somy
Park, Su-Jin
论文数: 0引用数: 0
h-index: 0
机构:
Korea Res Inst Biosci & Biotechnol, Funct Biomat Res Ctr, 181 Ipsin-gil, Jeongeup Si 56212, South KoreaChonnam Natl Univ, Res Inst Pharmaceut Sci, Coll Pharm, 77 Yongbong-ro, Gwangju 61186, South Korea
机构:
Natl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Taichung Vet Gen Hosp, Dept Phys Med & Rehabil, Taichung, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Cheng, Yuan-Yang
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Kao, Chung-Lan
Ma, Hsin-I
论文数: 0引用数: 0
h-index: 0
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Triserv Gen Hosp, Natl Def Med Ctr, Dept Neurol Surg, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Ma, Hsin-I
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Hung, Ching-Hsia
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Wang, Chin-Tien
Liu, Ding-Hao
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h-index: 0
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Natl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Taipei Vet Gen Hosp, Dept Phys Med & Rehabil, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
Liu, Ding-Hao
Chen, Po-Yin
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h-index: 0
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Taipei Vet Gen Hosp, Dept Phys Med & Rehabil, Taipei, TaiwanNatl Yang Ming Univ, Inst Clin Med, Taipei 112, Taiwan
机构:
Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Wang, Ning
Yu, Hai
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Yu, Hai
Song, Qian
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Song, Qian
Mao, Ping
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Mao, Ping
Li, Kuo
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h-index: 0
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
Li, Kuo
Bao, Gang
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Xi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R ChinaXi An Jiao Tong Univ, Affiliated Hosp 1, Dept Neurosurg, Xian 710061, Peoples R China
机构:
Olabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Alabi, Akinyinka O.
Ajayi, Abayomi M.
论文数: 0引用数: 0
h-index: 0
机构:
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Ajayi, Abayomi M.
Ben-Azu, Benneth
论文数: 0引用数: 0
h-index: 0
机构:
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, Nigeria
PAMO Univ Med Sci, Fac Basic Med Sci, Dept Pharmacol, Port Harcourt, Rivers State, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Ben-Azu, Benneth
Bakre, Adewale G.
论文数: 0引用数: 0
h-index: 0
机构:
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria
Bakre, Adewale G.
Umukoro, Solomon
论文数: 0引用数: 0
h-index: 0
机构:
Univ Ibadan, Neuropharmacol Unit, Dept Pharmacol & Therapeut, Fac Basic Med Sci,Coll Med, Ibadan, NigeriaOlabisi Onabanjo Univ, Fac Basic Med Sci, Dept Pharmacol & Therapeut, Ago Iwoye, Nigeria