New carborane-containing acids and amines

被引：16
作者：
Anufriev, S. A. [1 ]
Zakharova, M. V. [1 ]
Sivaev, I. B. [1 ]
Bregadze, V. I. [1 ]
机构：
[1] Russian Acad Sci, AN Nesmeyanov Inst Organoelement Cpds, 28 Ul Vavilova, Moscow 119991, Russia
来源：
RUSSIAN CHEMICAL BULLETIN | 2017年 / 66卷 / 09期
基金：
俄罗斯科学基金会;
关键词：
nido-carborane; sulfur-containing derivatives; amines; acids; NEUTRON-CAPTURE THERAPY; BRAIN-TUMORS; FUNCTIONAL-DERIVATIVES; CANCER; CHEMISTRY; DELIVERY;
D O I：
10.1007/s11172-017-1936-z
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Alkylation of nido-carborane methyl sulfide derivative [9-MeS-7,8-C2B9H11](-) was used to synthesize a series of new carborane-containing acids 9-HOOC(CH2) (n) (Me)S-7,8-C2B9H11 (n = 1-4) and amines 9-H2N(CH2) (n) (Me)S-7,8-C2B9H11 (n = 2, 3). The compounds obtained can be used for the development of BNCT agents.
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页码：1643 / 1649
页数：7
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