共 13 条
Consumption of high carbohydrate, high fat, and normal chow is equally suppressed by a cannabinoid receptor antagonist in non-deprived rats
被引:87
作者:

Verty, ANA
论文数: 0 引用数: 0
h-index: 0
机构: Univ New England, Sch Psychol, Armidale, NSW 2351, Australia

McGregor, IS
论文数: 0 引用数: 0
h-index: 0
机构: Univ New England, Sch Psychol, Armidale, NSW 2351, Australia

Mallet, PE
论文数: 0 引用数: 0
h-index: 0
机构:
Univ New England, Sch Psychol, Armidale, NSW 2351, Australia Univ New England, Sch Psychol, Armidale, NSW 2351, Australia
机构:
[1] Univ New England, Sch Psychol, Armidale, NSW 2351, Australia
[2] Univ Sydney, Sch Psychol, Sydney, NSW 2006, Australia
基金:
澳大利亚研究理事会;
关键词:
cannabinoid;
SR;
141716;
feeding;
rat;
D O I:
10.1016/j.neulet.2003.10.035
中图分类号:
Q189 [神经科学];
学科分类号:
071006 ;
摘要:
Administration of the CB1 receptor antagonist SR 141716 [N-piperidino-5-(4-chlorophenyl)- 1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide]. suppresses intake of highly palatable (high carbohydrate) food. However, the effects of SR 141716 on intake of foods with varying macronutrient compositions, and in non-deprived animals have not been well studied. In the present study, non-deprived rats were injected intraperitoneally with SR 141716 (0.03-3.0 mg/kg) and presented with a high carbohydrate, high fat, or normal chow diet. Food intake and locomotor activity were recorded for 120 min. Results showed that SR 141716 significantly suppressed food intake irrespective of the composition of the test food without affecting locomotor activity. These data suggest that food deprivation or high palatability of the ingesta are not necessary to observe the suppressive effects of SR 141716 on food intake. (C) 2003 Elsevier Ireland Ltd. All rights reserved.
引用
收藏
页码:217 / 220
页数:4
相关论文
共 13 条
[1]
Selective inhibition of sucrose and ethanol intake by SR 141716, an antagonist of central cannabinoid (CB1) receptors
[J].
Arnone, M
;
Maruani, J
;
Chaperon, F
;
Thiebot, MH
;
Poncelet, M
;
Soubrie, P
;
LeFur, G
.
PSYCHOPHARMACOLOGY,
1997, 132 (01)
:104-106

Arnone, M
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

Maruani, J
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

Chaperon, F
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

Thiebot, MH
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

Poncelet, M
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

Soubrie, P
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE

LeFur, G
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH,F-34084 MONTPELLIER,FRANCE
[2]
Involvement of central cannabinoid (CB1) receptors in the establishment of place conditioning in rats
[J].
Chaperon, F
;
Soubrié, P
;
Puech, AJ
;
Thiébot, MH
.
PSYCHOPHARMACOLOGY,
1998, 135 (04)
:324-332

Chaperon, F
论文数: 0 引用数: 0
h-index: 0
机构: Fac Med Pitie Salpetriere, INSERM U288, F-75634 Paris 13, France

Soubrié, P
论文数: 0 引用数: 0
h-index: 0
机构: Fac Med Pitie Salpetriere, INSERM U288, F-75634 Paris 13, France

Puech, AJ
论文数: 0 引用数: 0
h-index: 0
机构: Fac Med Pitie Salpetriere, INSERM U288, F-75634 Paris 13, France

Thiébot, MH
论文数: 0 引用数: 0
h-index: 0
机构: Fac Med Pitie Salpetriere, INSERM U288, F-75634 Paris 13, France
[3]
Leptin-regulated endocannabinoids are involved in maintaining food intake
[J].
Di Marzo, V
;
Goparaju, SK
;
Wang, L
;
Liu, J
;
Bátkai, S
;
Járai, Z
;
Fezza, F
;
Miura, GI
;
Palmiter, RD
;
Sugiura, T
;
Kunos, G
.
NATURE,
2001, 410 (6830)
:822-825

Di Marzo, V
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Goparaju, SK
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Wang, L
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Liu, J
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Bátkai, S
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Járai, Z
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Fezza, F
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Miura, GI
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Palmiter, RD
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Sugiura, T
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy

Kunos, G
论文数: 0 引用数: 0
h-index: 0
机构: CNR, Ist Chim Mol Interesse Biol, Endocannabinoid Res Grp, I-80072 Arco Felice Napoli, Naples, Italy
[4]
Effects of SR141716A, a central cannabinoid receptor antagonist, on food-maintained responding
[J].
Freedland, CS
;
Poston, JS
;
Porrino, LJ
.
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR,
2000, 67 (02)
:265-270

Freedland, CS
论文数: 0 引用数: 0
h-index: 0
机构:
Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA

Poston, JS
论文数: 0 引用数: 0
h-index: 0
机构:
Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA

Porrino, LJ
论文数: 0 引用数: 0
h-index: 0
机构:
Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA Wake Forest Univ, Bowman Gray Sch Med, Dept Physiol & Pharmacol, Winston Salem, NC 27157 USA
[5]
Cannabinoid influences on palatability:: microstructural analysis of sucrose drinking after Δ9-tetrahydrocannabinol, anandamide, 2-arachidonoyl glycerol and SR141716
[J].
Higgs, S
;
Williams, CM
;
Kirkham, TC
.
PSYCHOPHARMACOLOGY,
2003, 165 (04)
:370-377

Higgs, S
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Birmingham, Sch Psychol, Birmingham B15 2TT, W Midlands, England Univ Birmingham, Sch Psychol, Birmingham B15 2TT, W Midlands, England

Williams, CM
论文数: 0 引用数: 0
h-index: 0
机构: Univ Birmingham, Sch Psychol, Birmingham B15 2TT, W Midlands, England

Kirkham, TC
论文数: 0 引用数: 0
h-index: 0
机构: Univ Birmingham, Sch Psychol, Birmingham B15 2TT, W Midlands, England
[6]
Synergistic effects of opioid and cannabinoid antagonists on food intake
[J].
Kirkham, TC
;
Williams, CM
.
PSYCHOPHARMACOLOGY,
2001, 153 (02)
:267-270

Kirkham, TC
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reading, Dept Psychol, Reading RG6 6AL, Berks, England Univ Reading, Dept Psychol, Reading RG6 6AL, Berks, England

Williams, CM
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reading, Dept Psychol, Reading RG6 6AL, Berks, England Univ Reading, Dept Psychol, Reading RG6 6AL, Berks, England
[7]
Δ9-THC stimulates food intake in Lewis rats -: Effects on chow, high-fat and sweet high-fat diets
[J].
Koch, JE
.
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR,
2001, 68 (03)
:539-543

Koch, JE
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Wisconsin, Dept Psychol, Oshkosh, WI 54901 USA Univ Wisconsin, Dept Psychol, Oshkosh, WI 54901 USA
[8]
MODIFICATIONS OF NUTRIENT SELECTION INDUCED BY NALOXONE IN RATS
[J].
MARKSKAUFMAN, R
;
KANAREK, RB
.
PSYCHOPHARMACOLOGY,
1981, 74 (04)
:321-324

MARKSKAUFMAN, R
论文数: 0 引用数: 0
h-index: 0
机构:
TUFTS UNIV,DEPT PSYCHOL,MEDFORD,MA 02155 TUFTS UNIV,DEPT PSYCHOL,MEDFORD,MA 02155

KANAREK, RB
论文数: 0 引用数: 0
h-index: 0
机构:
TUFTS UNIV,DEPT PSYCHOL,MEDFORD,MA 02155 TUFTS UNIV,DEPT PSYCHOL,MEDFORD,MA 02155
[9]
Overeating, alcohol and sucrose consumption decrease in CB1 receptor deleted mice
[J].
Poncelet, M
;
Maruani, J
;
Calassi, R
;
Soubrié, P
.
NEUROSCIENCE LETTERS,
2003, 343 (03)
:216-218

Poncelet, M
论文数: 0 引用数: 0
h-index: 0
机构:
Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France

Maruani, J
论文数: 0 引用数: 0
h-index: 0
机构:
Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France

Calassi, R
论文数: 0 引用数: 0
h-index: 0
机构:
Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France

Soubrié, P
论文数: 0 引用数: 0
h-index: 0
机构:
Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France Sanofi Synthelabo Rech, Cent Nervous Syst Dept, F-34184 Montpellier 04, France
[10]
SR141716A, A POTENT AND SELECTIVE ANTAGONIST OF THE BRAIN CANNABINOID RECEPTOR
[J].
RINALDICARMONA, M
;
BARTH, F
;
HEAULME, M
;
SHIRE, D
;
CALANDRA, B
;
CONGY, C
;
MARTINEZ, S
;
MARUANI, J
;
NELIAT, G
;
CAPUT, D
;
FERRARA, P
;
SOUBRIE, P
;
BRELIERE, JC
;
LEFUR, G
.
FEBS LETTERS,
1994, 350 (2-3)
:240-244

RINALDICARMONA, M
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

BARTH, F
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

HEAULME, M
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

SHIRE, D
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

CALANDRA, B
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

CONGY, C
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

MARTINEZ, S
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

MARUANI, J
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

NELIAT, G
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

CAPUT, D
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

FERRARA, P
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

SOUBRIE, P
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

BRELIERE, JC
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE

LEFUR, G
论文数: 0 引用数: 0
h-index: 0
机构: SANOFI RECH, F-31676 LABEGE, FRANCE