Borrowing to make ends meet

被引:8
作者
Clardy, J [1 ]
机构
[1] Cornell Univ, Dept Chem & Biol Chem, Ithaca, NY 14853 USA
关键词
D O I
10.1073/pnas.96.5.1826
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1826 / 1827
页数:2
相关论文
共 11 条
[1]   Leukocyte protein tyrosine kinases: Potential targets for drug discovery [J].
Bolen, JB ;
Brugge, JS .
ANNUAL REVIEW OF IMMUNOLOGY, 1997, 15 :371-404
[2]   Affinity modulation of small-molecule ligands by borrowing endogenous protein surfaces [J].
Briesewitz, R ;
Ray, GT ;
Wandless, TJ ;
Crabtree, GR .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1999, 96 (05) :1953-1958
[3]   THE CHEMISTRY OF SIGNAL-TRANSDUCTION [J].
CLARDY, J .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1995, 92 (01) :56-61
[4]   Three-dimensional structure of the immunophilin-like domain of FKBP59 in solution [J].
Craescu, CT ;
Rouviere, N ;
Popescu, A ;
Cerpolini, E ;
Lebeau, MC ;
Baulieu, EE ;
Mispelter, J .
BIOCHEMISTRY, 1996, 35 (34) :11045-11052
[5]   DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS AND THE X-RAY CRYSTAL-STRUCTURES OF THEIR COMPLEXES WITH FKBP12 [J].
HOLT, DA ;
LUENGO, JI ;
YAMASHITA, DS ;
OH, HJ ;
KONIALIAN, AL ;
YEN, HK ;
ROZAMUS, LW ;
BRANDT, M ;
BOSSARD, MJ ;
LEVY, MA ;
EGGLESTON, DS ;
LIANG, J ;
SCHULTZ, LW ;
STOUT, TJ ;
CLARDY, J .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1993, 115 (22) :9925-9938
[6]   SH2 AND SH3 DOMAINS - ELEMENTS THAT CONTROL INTERACTIONS OF CYTOPLASMIC SIGNALING PROTEINS [J].
KOCH, CA ;
ANDERSON, D ;
MORAN, MF ;
ELLIS, C ;
PAWSON, T .
SCIENCE, 1991, 252 (5006) :668-674
[7]   PROTEIN MODULES AND SIGNALING NETWORKS [J].
PAWSON, T .
NATURE, 1995, 373 (6515) :573-580
[8]   CHEMISTRY AND BIOLOGY OF THE IMMUNOPHILINS AND THEIR IMMUNOSUPPRESSIVE LIGANDS [J].
SCHREIBER, SL .
SCIENCE, 1991, 251 (4991) :283-287
[9]   ATOMIC-STRUCTURE OF FKBP-FK506, AN IMMUNOPHILIN-IMMUNOSUPPRESSANT COMPLEX [J].
VANDUYNE, GD ;
STANDAERT, RF ;
KARPLUS, PA ;
SCHREIBER, SL ;
CLARDY, J .
SCIENCE, 1991, 252 (5007) :839-842
[10]   THE MECHANISM OF ACTION OF FK-506 AND CYCLOSPORINE-A [J].
WIEDERRECHT, G ;
LAM, E ;
HUNG, S ;
MARTIN, M ;
SIGAL, N .
IMMUNOSUPPRESSIVE AND ANTIINFLAMMATORY DRUGS, 1993, 696 :9-19