PET Imaging of CXCR4 Receptors in Cancer by a New Optimized Ligand

被引：160

作者：

Demmer, Oliver ^{[1
,2
]}

Gourni, Eleni ^{[3
]}

Schumacher, Udo ^{[4
]}

Kessler, Horst ^{[1
,2
,5
]}

Wester, Hans-Juergen ^{[3
]}

机构：

[1] Tech Univ Munich, Inst Adv Study, Dept Chem, D-85748 Garching, Germany

[2] Tech Univ Munich, Ctr Integrated Prot Sci, Dept Chem, D-85748 Garching, Germany

[3] Tech Univ Munich, Lehrstuhl Pharmazeut Radiochem, D-85748 Garching, Germany

[4] Univ Klinikum Hamburg Eppendorf, Inst Anat Expt Morphol 2, D-20246 Hamburg, Germany

[5] King Abdulaziz Univ, Fac Sci, Dept Chem, Jeddah 21589, Saudi Arabia

来源：

CHEMMEDCHEM | 2011年 / 6卷 / 10期

关键词：

CXCR4; DOTA; imaging agents; peptides; positron emission tomography; tracers; CHEMOKINE RECEPTOR; PERSONALIZED MEDICINE; HIGHLY POTENT; IN-VIVO; PEPTIDE; ANTAGONISTS; EXPRESSION; INHIBITOR; DISCOVERY; ONCOLOGY;

D O I：

10.1002/cmdc.201100320

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：1789 / 1791

页数：3

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