Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11b-hydroxysteroid dehydrogenase type 1 (11b-HSD1)

被引：0

作者：

Ye, Xiang-Yang ^{[1
]}

Chen, Stephanie Y. ^{[1
]}

Wu, Shung ^{[1
]}

Nayeem, Akbar ^{[2
]}

Yoon, David ^{[1
]}

Wang, Haixia ^{[1
]}

Hong, Zhenqiu ^{[1
]}

O'Connor, Steve ^{[1
]}

Apedo, Atsu ^{[3
]}

Li, James J. ^{[1
]}

Li, Jun ^{[1
]}

Kennedy, Lawrence ^{[1
]}

Walker, Steven ^{[1
]}

Golla, Rajasree ^{[4
]}

Seethala, Ramakrishna ^{[4
]}

Wang, Mengmeng ^{[5
]}

Harper, Timothy ^{[5
]}

Sleczka, Bogdan G.

Gordon, David ^{[6
]}

Robl, Jeffrey A. ^{[1
]}

机构：

[1] Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA

[2] Bristol Myers Squibb Co, CADD, Princeton, NJ 08543 USA

[3] Bristol Myers Squibb Co, DAS, Princeton, NJ 08543 USA

[4] Bristol Myers Squibb Co, Lead Evaluat, Princeton, NJ 08543 USA

[5] Bristol Myers Squibb Co, MAP, Princeton, NJ 08543 USA

[6] Bristol Myers Squibb Co, Dept Biol, Princeton, NJ 08543 USA

来源：

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2011年 / 242卷

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

138-MEDI

引用

页数：1

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