Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11b-hydroxysteroid dehydrogenase type 1 (11b-HSD1)

被引：0
作者：
Ye, Xiang-Yang [1 ]
Chen, Stephanie Y. [1 ]
Wu, Shung [1 ]
Nayeem, Akbar [2 ]
Yoon, David [1 ]
Wang, Haixia [1 ]
Hong, Zhenqiu [1 ]
O'Connor, Steve [1 ]
Apedo, Atsu [3 ]
Li, James J. [1 ]
Li, Jun [1 ]
Kennedy, Lawrence [1 ]
Walker, Steven [1 ]
Golla, Rajasree [4 ]
Seethala, Ramakrishna [4 ]
Wang, Mengmeng [5 ]
Harper, Timothy [5 ]
Sleczka, Bogdan G.
Gordon, David [6 ]
Robl, Jeffrey A. [1 ]
机构：
[1] Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA
[2] Bristol Myers Squibb Co, CADD, Princeton, NJ 08543 USA
[3] Bristol Myers Squibb Co, DAS, Princeton, NJ 08543 USA
[4] Bristol Myers Squibb Co, Lead Evaluat, Princeton, NJ 08543 USA
[5] Bristol Myers Squibb Co, MAP, Princeton, NJ 08543 USA
[6] Bristol Myers Squibb Co, Dept Biol, Princeton, NJ 08543 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2011年 / 242卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
138-MEDI
引用
收藏
页数：1
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