A novel linker strategy for solid-phase synthesis

被引：86

作者：

Morphy, JR ^{[1
]}

Rankovic, Z ^{[1
]}

Rees, DC ^{[1
]}

机构：

[1] ORGANON RES LABS LTD,DEPT MED CHEM,NEWHOUSE ML1 5SH,SCOTLAND

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 18期

关键词：

D O I：

10.1016/0040-4039(96)00497-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The REM resin for solid phase synthesis is described. Its use is illustrated by preparing a small array of tertiary amines using a Hofmann elimination reaction. No functional group is required for linking these compounds onto the resin other than the amine constructed during the synthesis. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：3209 / 3212

页数：4

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