Asymmetric synthesis of an aminomethyl morpholine via double allylic substitution

被引：43
|
作者：
Wilkinson, MC [1 ]
机构：
[1] GlaxoSmithKline, Chem Dev Div, Stevenage SG1 2NY, Herts, England
来源：
TETRAHEDRON LETTERS | 2005年 / 46卷 / 28期
关键词：
asymmetric synthesis; palladium; allylic substitution;
D O I：
10.1016/j.tetlet.2005.05.038
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The development of an asymmetric route to an aminomethyl morpholine intermediate via palladium-catalysed allylic substitution is described. (c) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码：4773 / 4775
页数：3
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