共 50 条
- [31] Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11b-hydroxysteroid dehydrogenase type 1 (11b-HSD1)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242Ye, Xiang-Yang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAChen, Stephanie Y.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAWu, Shung论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USANayeem, Akbar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, CADD, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAYoon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAWang, Haixia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAHong, Zhenqiu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAO'Connor, Steve论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAApedo, Atsu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, DAS, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USALi, James J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USALi, Jun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAKennedy, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAWalker, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAGolla, Rajasree论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Lead Evaluat, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USASeethala, Ramakrishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Lead Evaluat, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAWang, Mengmeng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, MAP, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAHarper, Timothy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, MAP, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USASleczka, Bogdan G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USAGordon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USARobl, Jeffrey A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Metab Dis Chem, Princeton, NJ 08543 USA
- [32] MEDI 334-Discovery, optimization and biological evaluation of novel, potent and selective histone deacetylase (HDAC) inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Namdev, Nivedita D.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USATandon, Manish论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAAkireddy, Rao论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAOrgueira, Hernan论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAVensel, David论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAKung, Ming论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAWu, Hui论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAHutchins, Patrick论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAMoussa, Magdi论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USALink, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USALiu, Yanbin论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USANicewonger, Robb论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USABruseo, Charles论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Mol Oncol, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAGorenstein, Julie论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Mol Oncol, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USANakuci, Enkeleda论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Mol Oncol, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAMcSweeney, Denise论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Mol Oncol, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USABresciano, Karen论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Preclin Dev, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAWang, Yunxia论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Preclin Dev, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAFrance, Dennis论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Mol Oncol, Woburn, MA 01801 USA ArQule Inc, Med Chem, Woburn, MA 01801 USAAshwell, Mark A.论文数: 0 引用数: 0 h-index: 0机构: ArQule Inc, Med Chem, Woburn, MA 01801 USA
- [33] Synthesis and biological evaluation of picolinamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (03) : 695 - 700Ryu, Je Ho论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 151742, South Korea Seoul Natl Univ, Coll Pharm, Seoul 151742, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaKim, Shinae论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaHan, Hye Young论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaSon, Hyun Joo论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaLee, Hyun Jung论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaShin, Young Ah论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaKim, Jae-Sun论文数: 0 引用数: 0 h-index: 0机构: SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South KoreaPark, Hyeung-geun论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 151742, South Korea Seoul Natl Univ, Coll Pharm, Seoul 151742, South Korea SK Chem, Life Sci R&D Ctr, Songnam 463400, South Korea
- [34] Identification of adamantyl urea derivatives as novel and selective 11β-HSD1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Fujiwara, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanSuda, Hitoshi论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanNishimura, Tamiki论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanNunami, Noriko论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanSato, Yasuhiro论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Genom Sci Res, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanNegishi, Toru论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacokinet Res, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanHiramine, Yasushi论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol Res, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanKohayakawa, Chie论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol Res, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, JapanHoriuchi, Yoshihiro论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem Resarch, Suita, Osaka 5640053, Japan
- [35] Optimization of 1,2,4-triazolopyridines as inhibitors of human 11β-hydroxysteroid dehydrogenase Type 1 (11β-HSD-1): Discovery of clinical candidate BMS-823778ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250Li, Jun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAKennedy, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAWang, Haixia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USALi, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAWalker, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAHong, Zhenqiu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAO'Connor, Stephen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAYe, Xiang-Yang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAChen, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAWu, Shung论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAYoon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USANayeem, Akbar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USACamac, Daniel论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAMorin, Paul论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USASheriff, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAWang, Mengmeng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAHarper, Tim论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAGolla, Rajasree论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USASeethala, Ramakrishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAHarrity, Thomas论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAPonticiello, Randolph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAMorgan, Nathan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USATaylor, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAZebo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USAGordon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USARobl, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Pennington, NJ USA Bristol Myers Squibb, Pennington, NJ USA
- [36] Discovery of novel sulfonamides as potent and selective inhibitors against human and mouse 11β-hydroxysteroid dehydrogenase type 1MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2012, 358 (01) : 46 - 52Xia, Guangxin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLiu, Lin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaXue, Mengzhu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLiu, Haiyan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaYu, Jianxin论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLi, Ping论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaChen, Qian论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaXiong, Bing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLiu, Xuejun论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaShen, Jingkang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China
- [37] Efficacy and safety of the selective 11β-HSD-1 inhibitors MK-0736 and MK-0916 in overweight and obese patients with hypertensionJOURNAL OF THE AMERICAN SOCIETY OF HYPERTENSION, 2011, 5 (03) : 166 - 176Shah, Sukrut论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAHermanowski-Vosatka, Anne论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAGibson, Kendra论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USARuck, Rae Ann论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAJia, Gang论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAZhang, John论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAHwang, Peggy M. T.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USARyan, Nicholas W.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USALangdon, Ronald B.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USAFeig, Peter U.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA Merck Sharp & Dohme Corp, Rahway, NJ 07065 USA
- [38] Discovery of Novel 11β-HSD1 Inhibitors by Pharmacophore-Based Virtual ScreeningBULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2012, 33 (07) : 2365 - 2368Kim, Nam Doo论文数: 0 引用数: 0 h-index: 0机构: YOUAI Co Ltd, R&D Ctr, Suwon 443766, South Korea Univ Incheon, Div Life Sci, Inchon 406772, South KoreaLee, Younho论文数: 0 引用数: 0 h-index: 0机构: YOUAI Co Ltd, R&D Ctr, Suwon 443766, South Korea Univ Incheon, Div Life Sci, Inchon 406772, South KoreaHan, Chang-Kyun论文数: 0 引用数: 0 h-index: 0机构: Ahn Gook Pharm, R&D Ctr, Suwon 443766, South Korea Univ Incheon, Div Life Sci, Inchon 406772, South KoreaAhn, Soon Kil论文数: 0 引用数: 0 h-index: 0机构: Univ Incheon, Div Life Sci, Inchon 406772, South Korea Univ Incheon, Div Life Sci, Inchon 406772, South Korea
- [39] Discovery and optimization of piperidyl benzamide derivatives as a novel class of 11β-HSD1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (06) : 1797 - 1801Rew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAMcMinn, Dustin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAWang, Zhulun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAHe, Xiao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAHungate, Randall W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAJaen, Juan C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASudom, Athena论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USATu, Hua论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAUrsu, Stefania论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAVillemure, Elisia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAWalker, Nigel P. C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAPowers, Jay P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USA
- [40] Discovery of benzoylpiperazines as a novel class of potent and selective GlyT1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (18) : 5134 - 5139Pinard, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandAlberati, Daniela论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CNS Dis Biol Area, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandBorroni, Edilio论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CNS Dis Biol Area, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandFischer, Holger论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandHainzl, Dominik论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Non Clin Safety, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandJolidon, Synese论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandMoreau, Jean-Luc论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CNS Dis Biol Area, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandNarquizian, Robert论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandNettekoven, Matthias论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandNorcross, Roger D.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandStalder, Henri论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, SwitzerlandThomas, Andrew W.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, Discovery Chem, CH-4070 Basel, Switzerland