Design, synthesis and antimycotic activity of (N-heteroaryl)aryemethanamines

被引:0
|
作者
Ballistreri, A
Bottino, A
Musumarra, G
Fioravanti, R
Biava, M
Porretta, GC
Simonetti, N
Villa, A
机构
[1] UNIV CATANIA,DIPARTIMENTO SCI CHIM,I-95125 CATANIA,ITALY
[2] UNIV ROMA LA SAPIENZA,DIPARTIMENTO STUDI CHIM TECNOL SOSTANCE BIOL ATT,I-00185 ROME,ITALY
[3] UNIV ROMA LA SAPIENZA,IST MICROBIOL,I-00185 ROME,ITALY
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The design, synthesis and antimycotic activities of 18 (N-heteroaryl)arylmethanamines are reported. The MIC against Candida strains of the most active amine, 3-(p-methylbenzylamino)quinoline, is comparable to that of pyrrolnitrin.
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页码:61 / 65
页数:5
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