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- [22] ACTIVITY OF MLN4924, A NOVEL FIRST IN CLASS SMALL MOLECULE INHIBITOR OF THE NEDD8 ACTIVATING ENZYME, IN PRECLINICAL MODELS OF ACUTE MYELOID LEUKEMIAHAEMATOLOGICA-THE HEMATOLOGY JOURNAL, 2009, 94 : 305 - 306Swords, T.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USAKelly, K.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USASmith, P.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USAMahalingam, D.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USAO'Dwyer, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Coll Hosp Galway, Galway, Ireland Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USANawrocki, S.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USAGiles, F.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USACarew, J.论文数: 0 引用数: 0 h-index: 0机构: Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA Canc Therapy & Res Ctr S Texas, San Antonio, TX 78229 USA
- [23] Radiosensitization of Human Pancreatic Cancer Cells by MLN4924, an Investigational NEDD8-Activating Enzyme InhibitorCANCER RESEARCH, 2012, 72 (01) : 282 - 293Wei, Dongping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALi, Hua论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAYu, Jie论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASebolt, Jonathan T.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAZhao, Lili论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALawrence, Theodore S.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAMorgan, Meredith A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASun, Yi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA
- [24] Targeting protein neddylation with an NEDD8-activating enzyme inhibitor MLN4924 induced apoptosis or senescence in human lymphoma cellsCANCER BIOLOGY & THERAPY, 2015, 16 (03) : 420 - 429Wang, Yanchun论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R China Fudan Univ, Sch Basic Med Sci, Dept Immunol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaLuo, Zhongguang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Basic Med Sci, Dept Immunol, Shanghai 200433, Peoples R China Fudan Univ, Huashan Hosp, Dept Digest Dis, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaPan, Yongfu论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Basic Med Sci, Dept Immunol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaWang, Weige论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Dept Pathol,Dept Oncol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaZhou, Xiaoyan论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Dept Pathol,Dept Oncol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaJeong, Lak Shin论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Coll Pharm, Seoul, South Korea Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaChu, Yiwei论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Basic Med Sci, Dept Immunol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaLiu, Jie论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Basic Med Sci, Dept Immunol, Shanghai 200433, Peoples R China Fudan Univ, Huashan Hosp, Dept Digest Dis, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R ChinaJia, Lijun论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R China Fudan Univ, Shanghai Med Coll, Shanghai Canc Ctr, Canc Inst,Dept Oncol, Shanghai 200433, Peoples R China
- [25] Initial testing of the investigational NEDD8-activating enzyme inhibitor MLN4924 by the pediatric preclinical testing programPEDIATRIC BLOOD & CANCER, 2012, 59 (02) : 246 - 253Smith, Malcolm A.论文数: 0 引用数: 0 h-index: 0机构: NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAMaris, John M.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Childrens Hosp Philadelphia, Sch Med, Philadelphia, PA 19104 USA Abramson Family Canc Res Inst, Philadelphia, PA USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAGorlick, Richard论文数: 0 引用数: 0 h-index: 0机构: Childrens Hosp Montefiore, Bronx, NY USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAKolb, E. Anders论文数: 0 引用数: 0 h-index: 0机构: Alfred I DuPont Hosp Children, Wilmington, DE USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USALock, Richard论文数: 0 引用数: 0 h-index: 0机构: Childrens Canc Inst Australia Med Res, Randwick, NSW, Australia NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USACarol, Hernan论文数: 0 引用数: 0 h-index: 0机构: Childrens Canc Inst Australia Med Res, Randwick, NSW, Australia NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAKeir, Stephen T.论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Med Ctr, Durham, NC USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAReynolds, C. Patrick论文数: 0 引用数: 0 h-index: 0机构: Texas Tech Univ, Hlth Sci Ctr, Lubbock, TX 79430 USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAKang, Min H.论文数: 0 引用数: 0 h-index: 0机构: Texas Tech Univ, Hlth Sci Ctr, Lubbock, TX 79430 USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAMorton, Christopher L.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Memphis, TN 38105 USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAWu, Jianrong论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Memphis, TN 38105 USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAYu, Jie论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USAHoughton, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USA
- [26] Quantifiable analysis of cellular pathway inhibition of a Nedd8-activating enzyme inhibitor, MLN4924, using AlphaScreenANALYTICAL BIOCHEMISTRY, 2013, 439 (02) : 109 - 115Yan, Zhong-Hua论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABurkhardt, Anne论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USALoke, Huay-Keng论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAChen, Jesse论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAXu, Qing论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABrauer, Pam论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAMa, Jingya论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USALin, Yafang论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAGarcia, Khris论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USADick, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABembenek, Michael E.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USA
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