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- [21] The selective 5-HT2A receptor agonist 25CN-NBOH: Structure-activity relationship, in vivo pharmacology, and in vitro and ex vivo binding characteristics of [3H]25CN-NBOHBIOCHEMICAL PHARMACOLOGY, 2020, 177Jensen, Anders A.Halberstadt, Adam L.Marcher-Rorsted, EmilOdland, Anna U.Chatha, MuhammadSpeth, NikolajLiebscher, GudrunHansen, MartinBrauner-Osborne, HansPalner, MikaelAndreasen, Jesper T.Kristensen, Jesper L.
- [22] In vivo and in vitro ADMET profiling and in vivo pharmacodynamic investigations of a selective α7 nicotinic acetylcholine receptor agonist with a spirocyclic Δ2-isoxazoline molecular skeletonEUROPEAN JOURNAL OF PHARMACOLOGY, 2018, 820 : 265 - 273Matera, CarloDondio, GiulioBraida, DanielaPonzoni, LuisaDe Amici, MarcoSala, MariaelvinaDallanoce, Clelia
- [23] Novel, Selective Inhibitors of USP7 Uncover Multiple Mechanisms of Antitumor Activity In Vitro and In VivoMOLECULAR CANCER THERAPEUTICS, 2020, 19 (10) : 1970 - 1980Ohol, Yamini M.Sun, Michael T.Cutler, GeneLeger, Paul R.Hu, Dennis X.Biannic, BerengerRana, PayalCho, CynthiaJacobson, ScottWong, Steve T.Sanchez, JerickShah, NiketPookot, DeepaAbraham, BettyYoung, KyleSuthram, SilpaMarshall, Lisa A.Bradford, DeliaKozon, NathanHan, XinpingOkano, AkinoriMaung, JackColas, ChristopheSchwarz, JacobWustrow, DavidBrockstedt, Dirk G.Kassner, Paul D.
- [24] Discovery of potent and selective inhibitors of USP7 with anti-tumor activity in vitro and in vivoCANCER RESEARCH, 2019, 79 (13)Ohol, Yamini M.Sun, MichaelLeger, PaulHu, DennisBiannic, BerengerRana, PayalCho, CynthiaJacobson, ScottWong, SteveSanchez, JerickHan, XinpingYoung, KyleOkano, AkinoriMaung, JackCutler, GeneShah, NickAdusumilli, LavanyaKaveri, DeepikaTalay, OezcanPookot, DeepaAbraham, BettyBradford, DeliaKozon, NathanColas, ChristopheKim, AndreaSchwarz, JacobWustrow, DavidBrockstedt, DirkKassner, Paul
- [25] The in vivo -: Preclinical profile of TD-5108, a selective, high intrinsic activity 5-HT4 receptor agonistGASTROENTEROLOGY, 2007, 132 (04) : A688 - A688Beattie, David T.Armstrong, Scott R.Marquess, DanielShaw, Jeng-PengSmith, Jacqueline A.Humphrey, Patrick P.
- [26] Structure-activity relationship, in vitro and in vivo evaluation of novel dienyl sulphonyl fluorides as selective BuChE inhibitors for the treatment of Alzheimer's diseaseJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2021, 36 (01) : 1860 - 1873Wu, ChengyaoZhang, GuijuanZhang, Zai-WeiJiang, XiaZhang, ZiwenLi, HuanhuanQin, Hua-LiTang, Wenjian
- [27] The copper(II) complexes of new anthrahydrazone ligands: In vitro and in vivo antitumor activity and structure-activity relationshipJOURNAL OF INORGANIC BIOCHEMISTRY, 2020, 212Liu, Rui-XueWang, Chen-YuWu, Ying-ShuLuo, Ru-YiJiang, Xiao-HongTang, Meng-TingLiu, Yan-ChengChen, Zhen-FengLiang, Hong
- [28] The in vitro pharmacological profile of TD-5108, a selective 5-HT4 receptor agonist with high intrinsic activityNAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2008, 378 (01) : 125 - 137Smith, J. A. M.Beattie, D. T.Marquess, D.Shaw, J. -P.Vickery, R. G.Humphrey, P. P. A.
- [29] The in vitro pharmacological profile of TD-5108, a selective 5-HT4 receptor agonist with high intrinsic activityNaunyn-Schmiedeberg's Archives of Pharmacology, 2008, 378 : 125 - 137J. A. M. SmithD. T. BeattieD. MarquessJ.-P. ShawR. G. VickeryP. P. A. Humphrey
- [30] Development of a potent and selective GPR7 agonist: A systematic structure-activity study of neuropeptide BNEUROSCIENCE RESEARCH, 2007, 58 : S76 - S76Kanesaka, MakiMatsuda, MasaoHirano, AtsushiTanaka, KenichiKanatani, AkioTokita, Shigeru