Synthesis and structure characterization of two thienonaphthopyrones

被引：0

作者：

Fan, MC ^{[1
]}

Qian, XH

Tao, ZF

机构：

[1] Sichuan Inst Light Ind & Chem Tech, Dept Chem Engn, Zigong 643033, Peoples R China

[2] E China Univ Sci & Technol, Inst Pesticides & Pharmaceut, Shanghai 200237, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2000年 / 20卷 / 03期

关键词：

thienonaphthopyrone; synthesis; X - ray crystal structure; characterization;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Two novel angular thienonaphthopyrones 6 and 8 were synthesized starting from 2,7 - naphthalenediol in six steps, respectively. The crystal structure of 6 was determined. The planarity of 6 and the geometry of the active double bond between the alpha - pyrone and the thieno moieties of 6 suggest that thienonaphthopyrones might be useful as efficient monofunctional DNA intercalators.

引用

页码：338 / 343

页数：6

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