Synthesis of some novel functionalized dihydropyrido[2,3-d]pyrimidines via an one-pot three-component reaction catalysed by InCl3

被引:28
作者
Naidu, P. Seetham [1 ]
Borah, Pallabi [1 ]
Bhuyan, Pulak J. [1 ]
机构
[1] CSIR NE Inst Sci & Technol, Div Med Chem, Jorhat 785006, Assam, India
关键词
Dihydropyridine; Pyrimidine; Indole; Multi-component reactions (MCRs); Indium chloride; THIOPYRANO INDOLE-DERIVATIVES; POLYHYDROQUINOLINE DERIVATIVES; SIMPLE OXINDOLE; FACILE; ANALOGS; COMPLEX;
D O I
10.1016/j.tetlet.2012.05.102
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Some novel functionalized dihydropyrido[2,3-d]pyrimidine derivatives 4 were synthesized using a one-pot three-component reaction of 6-aminouracils 1, aryl aldehydes 2 and 3-cyanoacetyl indole 3 using InCl3 as catalyst. (C) 2012 Elsevier Ltd. All rights reserved.
引用
收藏
页码:4015 / 4017
页数:3
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