2-amino-2-oxazolines, part 9:: Synthesis and pharmacological evaluation of N-phenyl-N′-[1-[3-(1-aryl-4-piperazinyl)propan-2-ol]]ureas

被引：0
|
作者：
Bosc, JJ [1 ]
Jarry, C [1 ]
机构：
[1] Univ Bordeaux 2, UFR Sci Pharmaceut, Chim Phys Lab, F-33076 Bordeaux, France
来源：
ARCHIV DER PHARMAZIE | 1998年 / 331卷 / 09期
关键词：
2-amino-2-oxazoline; 3-phenylcarbamoyl-2-iminooxazolidine; N-phenyl-N '-[l-[3-(1-aryl-4-piperazinyl)-propan-2-ol]]urea; antiallergic and analgesic activities;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
N-Phenyl-N'-[1-[3-(1-aryl-4-piperazinyl)propan-2-ol]]ureas (3) were synthesized from the 3-phenylcarbamoyl-5-[( 1-aryl-4-piperazinyl)methyl]-2-iminooxazolidines (1) via the corresponding 2-oxazolidinones (2). The prepared compounds were screened for their antiallergic and analgesic activities.
引用
收藏
页码：291 / 293
页数：3
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