A general and convenient synthesis of N-aryl piperazines

被引:61
作者
Liu, KG [1 ]
Robichaud, AJ [1 ]
机构
[1] Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USA
关键词
N-aryl piperazines;
D O I
10.1016/j.tetlet.2005.09.092
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A general and convenient synthesis of N-aryl piperazines from bis(2-chloroethyl)amine hydrochloride and a broad range of anilines in diethylene glycol monomethyl ether is described. (c) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码:7921 / 7922
页数:2
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