Unique general anesthetic binding sites within distinct conformational states of the nicotinic acetylcholine receptor

被引:61
作者
Arias, HR [1 ]
Kem, WR
Trudell, JR
Blanton, MP
机构
[1] Western Univ Hlth Sci, Coll Pharm, Dept Pharmaceut Sci, Pomona, CA 91766 USA
[2] Univ Florida, Coll Med, Dept Pharmacol & Therapeut, Gainesville, FL 32610 USA
[3] Stanford Univ, Sch Med, Dept Anesthesia, Stanford, CA 94305 USA
[4] Texas Tech Univ, Hlth Sci Ctr, Sch Med, Dept Pharmacol, Lubbock, TX 79430 USA
[5] Texas Tech Univ, Hlth Sci Ctr, Sch Med, Dept Anesthesiol, Lubbock, TX 79430 USA
来源
INTERNATIONAL REVIEW OF NEUROBIOLOGY, VOL 54 | 2003年 / 54卷
关键词
D O I
10.1016/S0074-7742(03)54002-8
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:1 / 52
页数:52
相关论文
共 224 条
[11]   Characterization of the dizocilpine binding site on the nicotinic acetylcholine receptor [J].
Arias, HR ;
Mccardy, EA ;
Blanton, MP .
MOLECULAR PHARMACOLOGY, 2001, 59 (05) :1051-1060
[12]   5-doxylstearate-induced displacement of phencyclidine from its low-affinity binding sites on the nicotinic acetylcholine receptor [J].
Arias, HR .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1999, 371 (01) :89-97
[13]  
Arias HR, 2001, MOL PHARMACOL, V60, P497
[14]   QUINACRINE AND ETHIDIUM BIND TO DIFFERENT LOCI ON THE TORPEDO ACETYLCHOLINE-RECEPTOR [J].
ARIAS, HR ;
VALENZUELA, CF ;
JOHNSON, DA .
BIOCHEMISTRY, 1993, 32 (24) :6237-6242
[15]   Role of local anesthetics on both cholinergic and serotonergic ionotropic receptors [J].
Arias, HR .
NEUROSCIENCE AND BIOBEHAVIORAL REVIEWS, 1999, 23 (06) :817-843
[16]  
ARIAS HR, 1993, J BIOL CHEM, V268, P6348
[17]  
ARIAS HR, 2002, IN PRESS RECENT RES
[18]  
ARIAS HR, 2002, UNPUB BIOCHEMISTRY
[19]  
ARIAS HR, 2001, DRUG RECEPTOR THERMO, P293
[20]   ACTION OF ENFLURANE ON CHOLINERGIC TRANSMISSION IN IDENTIFIED APLYSIA NEURONS [J].
ARIMURA, H ;
IKEMOTO, Y .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 89 (03) :573-582