共 50 条
- [1] Discovery of selective inhibitors of mutant b-rafABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 237Deal, Judith G.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAPalmer, Cynthia L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USARomines, William H.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAPark, Julie Y.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAGuo, Lisa C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAZehnder, Luke论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAMarrone, Tami J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAMcTigue, Michele论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USADeLisle, Dorothy论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USASolowiej, James论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USAYu, Xiao-Hong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USABagrodia, Shubha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA Pfizer Global Res & Dev La Jolla, San Diego, CA 92121 USA
- [2] Discovery of potent, selective inhibitors of mutant B-RafABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242Palmer, Cynthia L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USACui, Jingrong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USADeal, Judith论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAGu, Danlin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAGuo, Chuangxing论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAKephart, Susan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USALinton, Maria A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAMcAlpine, Indrawan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAPairish, Mason论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USABagrodia, Shubha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USACao, Yixue论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAYamazaki, Shinji论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USADeLisle, Dorothy论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USAJohn-Baptiste, Annette论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, San Diego, CA 92121 USA
- [3] Mutant B-Raf Kinase Inhibitors as Anticancer AgentsANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 2016, 16 (12) : 1558 - 1575Asati, Vivek论文数: 0 引用数: 0 h-index: 0机构: Guru Ghasidas Vishwavidyalaya, Inst Pharmaceut Sci, Bilaspur 495009, Chhattisgarh, India Guru Ghasidas Vishwavidyalaya, Inst Pharmaceut Sci, Bilaspur 495009, Chhattisgarh, IndiaBharti, Sanjay K.论文数: 0 引用数: 0 h-index: 0机构: Guru Ghasidas Vishwavidyalaya, Inst Pharmaceut Sci, Bilaspur 495009, Chhattisgarh, India Guru Ghasidas Vishwavidyalaya, Inst Pharmaceut Sci, Bilaspur 495009, Chhattisgarh, IndiaMahapatra, Debarshi K.论文数: 0 引用数: 0 h-index: 0机构: Indian Inst Chem Technol, Nat Prod Chem Div, Genet Chem Lab, CSIR, Hyderabad 500007, Telangana, India Guru Ghasidas Vishwavidyalaya, Inst Pharmaceut Sci, Bilaspur 495009, Chhattisgarh, India
- [4] Non-oxime pyrazole based inhibitors of B-Raf kinaseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (11) : 3488 - 3492Newhouse, Bradley J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAHansen, Joshua D.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAWelch, Mike论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USATopalov, George论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USALittman, Nicole论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USACallejo, Michele论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAGalbraith, Sarah论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USALaird, Ellen R.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USABrandhuber, Barbara J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAVigers, Guy论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAMorales, Tony论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USAWoessner, Rich论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USARandolph, Nikole论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Array BioPharma, Boulder, CO 80301 USALyssikatos, Joseph论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma, Boulder, CO 80301 USAOlivero, Alan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma, Boulder, CO 80301 USA
- [5] Potent and selective pyrazole-based inhibitors of B-Raf kinaseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (16) : 4692 - 4695Hansen, Joshua D.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USANewhouse, Brad论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAWelch, Mike论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USATopalov, George论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USALittman, Nicole论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USACallejo, Michele论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAGloor, Susan论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USALaird, Ellen论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USABrandhuber, Barbara J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAVigers, Guy论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAMorales, Tony论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAWoessner, Rich论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USARandolph, Nikole论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USALyssikatos, Joseph论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USAOlivero, Alan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma, Lead Optimizat, Boulder, CO 80301 USA
- [6] Autophagy-Dependent Survival of Mutant B-Raf Melanoma Cells Selected for Resistance to Apoptosis Induced by Inhibitors against Oncogenic B-RafBIOMOLECULES & THERAPEUTICS, 2013, 21 (02) : 114 - 120Ahn, Jun-Ho论文数: 0 引用数: 0 h-index: 0机构: Univ lncheon, Coll Life Sci & Bioengn, Div Life Sci, Inchon 406772, South Korea Univ lncheon, Coll Life Sci & Bioengn, Div Life Sci, Inchon 406772, South KoreaLee, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ lncheon, Coll Life Sci & Bioengn, Div Life Sci, Inchon 406772, South Korea Univ lncheon, Coll Life Sci & Bioengn, Div Life Sci, Inchon 406772, South Korea
- [7] B-Raf and the inhibitors: from bench to bedsideJournal of Hematology & Oncology, 6Tiangui Huang论文数: 0 引用数: 0 h-index: 0机构: Westchester Medical Center and New York Medical College,Department of PathologyMichael Karsy论文数: 0 引用数: 0 h-index: 0机构: Westchester Medical Center and New York Medical College,Department of PathologyJian Zhuge论文数: 0 引用数: 0 h-index: 0机构: Westchester Medical Center and New York Medical College,Department of PathologyMinghao Zhong论文数: 0 引用数: 0 h-index: 0机构: Westchester Medical Center and New York Medical College,Department of PathologyDelong Liu论文数: 0 引用数: 0 h-index: 0机构: Westchester Medical Center and New York Medical College,Department of Pathology
- [8] B-Raf kinase inhibitors for cancer treatmentCURRENT OPINION IN INVESTIGATIONAL DRUGS, 2007, 8 (06) : 452 - 456Li, Nanxin论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USABatt, David论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAWarmuth, Markus论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA
- [9] Selective Inhibitors of the Mutant B-Raf Pathway: Discovery of a Potent and Orally Bioavailable AminoisoquinolineJOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (20) : 6189 - 6192Smith, Adrian L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USADeMorin, Frenel F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAParas, Nick A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHuang, Qi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAPetkus, Jeffrey K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USADoherty, Elizabeth M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USANixey, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAKim, Joseph L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAWhittington, Douglas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAEpstein, Linda F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USALee, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USARose, Mark J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USABabij, Carol论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAFernando, Manory论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHess, Kristen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USALe, Quynh论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USABeltran, Pedro论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USACarnahan, Josette论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA
- [10] Development of potent inhibitors of B-Raf kinaseABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Wei, Jianmei论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, San Diego, CA 92121 USA Johnson & Johnson Pharmaceut Res & Dev LLC, San Diego, CA 92121 USAWolin, Ronald论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, San Diego, CA 92121 USA Johnson & Johnson Pharmaceut Res & Dev LLC, San Diego, CA 92121 USA