Trifluoromethylation of aryl and heteroaryl halides

被引：286
|
作者：
Roy, Sudipta [1 ]
Gregg, Brian T. [1 ]
Gribble, Gordon W. [2 ]
Le, Van-Duc [1 ]
Roy, Sujata [1 ]
机构：
[1] AMRI, Dept Med Chem, 26 Corp Circle, Albany, NY 12212 USA
[2] Dartmouth Coll, Dept Chem, Hanover, NH 03755 USA
来源：
TETRAHEDRON | 2011年 / 67卷 / 12期
关键词：
CROSS-COUPLING REACTIONS; PHENYLETHANOLAMINE N-METHYLTRANSFERASE; FORMING REDUCTIVE ELIMINATION; ORGANIC FLUORINE-COMPOUNDS; NUCLEOPHILIC TRIFLUOROMETHYLATION; MEDICINAL CHEMISTRY; 1-AND 2-(TRIFLUOROMETHYL)NAPHTHALENES; BIOLOGICAL EVALUATION; SELECTIVE INHIBITORS; SYNTHETIC METHODS;
D O I：
10.1016/j.tet.2011.01.002
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[No abstract available]
引用
收藏
页码：2161 / 2195
页数：35
相关论文
共 50 条
  • [31] Ambient temperature, Ullmann-like reductive coupling of aryl, heteroaryl, and alkenyl halides
    Zhang, SJ
    Zhang, DW
    Liebeskind, LS
    JOURNAL OF ORGANIC CHEMISTRY, 1997, 62 (08): : 2312 - 2313
  • [32] Triton B-Mediated Efficient and Convenient Alkoxylation of Activated Aryl and Heteroaryl Halides
    Meshram, H. M.
    Goud, P. Ramesh
    Reddy, B. Chennakesava
    Kumar, D. Aravind
    SYNTHETIC COMMUNICATIONS, 2010, 40 (14) : 2122 - 2129
  • [33] Negishi cross-coupling of secondary alkylzinc halides with aryl/heteroaryl halides using Pd-PEPPSI-IPent
    Calimsiz, Selcuk
    Organ, Michael G.
    CHEMICAL COMMUNICATIONS, 2011, 47 (18) : 5181 - 5183
  • [34] A general synthesis of a-aryl and heteroarylpyrroles by palladium-catalyzed coupling reaction of a-tributylstannylpyrrole with aryl and heteroaryl halides
    Wang, J.
    Scott, A. I.
    Tetrahedron Letters, 37 (19):
  • [35] Coupling of organotin reagents with aryl, acyl and heteroaryl halides .2. Synthesis of thienylpyridine derivatives
    Sosabowski, MH
    Powell, P
    JOURNAL OF CHEMICAL RESEARCH-S, 1997, (01): : 12 - 13
  • [36] Iron-Catalyzed Cross-Coupling of Benzylic Manganese Chlorides with Aryl and Heteroaryl Halides
    Benischke, Andreas D.
    Breuillac, Antoine J. A.
    Moyeux, Alban
    Cahiez, Gerard
    Knochel, Paul
    SYNLETT, 2016, 27 (03) : 471 - 476
  • [37] C-O Cross-Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols
    Maligres, Peter E.
    Li, Jing
    Krska, Shane W.
    Schreier, John D.
    Raheem, Izzat T.
    ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2012, 51 (36) : 9071 - 9074
  • [38] Solvent-Free Buchwald-Hartwig Reaction of Aryl and Heteroaryl Halides with Secondary Amines
    Topchiy, Maxim A.
    Asachenko, Andrey F.
    Nechaev, Mikhail S.
    EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2014, 2014 (16) : 3319 - 3322
  • [39] Palladium-Catalyzed N-Arylation of Iminodibenzyls and Iminostilbenes with Aryl-and Heteroaryl Halides
    Huang, Wenliang
    Buchwald, Stephen L.
    CHEMISTRY-A EUROPEAN JOURNAL, 2016, 22 (40) : 14186 - 14189
  • [40] Visible light-induced aryltrifluoromethylation of hydroxy alkenes via radical trifluoromethylation-triggered aryl and heteroaryl migration
    Wang, Hao
    Xu, Qian
    Yu, Shouyun
    ORGANIC CHEMISTRY FRONTIERS, 2018, 5 (14): : 2224 - 2228
12345