Trifluoromethylation of aryl and heteroaryl halides

被引：286

作者：

Roy, Sudipta ^{[1
]}

Gregg, Brian T. ^{[1
]}

Gribble, Gordon W. ^{[2
]}

Le, Van-Duc ^{[1
]}

Roy, Sujata ^{[1
]}

机构：

[1] AMRI, Dept Med Chem, 26 Corp Circle, Albany, NY 12212 USA

[2] Dartmouth Coll, Dept Chem, Hanover, NH 03755 USA

来源：

TETRAHEDRON | 2011年 / 67卷 / 12期

关键词：

CROSS-COUPLING REACTIONS; PHENYLETHANOLAMINE N-METHYLTRANSFERASE; FORMING REDUCTIVE ELIMINATION; ORGANIC FLUORINE-COMPOUNDS; NUCLEOPHILIC TRIFLUOROMETHYLATION; MEDICINAL CHEMISTRY; 1-AND 2-(TRIFLUOROMETHYL)NAPHTHALENES; BIOLOGICAL EVALUATION; SELECTIVE INHIBITORS; SYNTHETIC METHODS;

D O I：

10.1016/j.tet.2011.01.002

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：2161 / 2195

页数：35

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