SYNTHESIS AND BIOEFFICACY TEST OF SOME NOVEL HALOGENATED-4-[(SUBSTITUTED-BENZOTHIAZOL-2-YL)-HYDRAZONO]-2-(SUBSTITUTED PHENYL)-5-METHYL-2, 4-DIHYDRO-PYRAZOL-3-ONE

被引：6

作者：

Sareen, V. ^{[1
]}

Khatri, V. ^{[1
]}

Sharma, K. ^{[1
]}

Shinde, D. ^{[1
]}

Sareen, S. ^{[1
]}

机构：

[1] Univ Rajasthan, Dept Chem, Jaipur 302004, Rajasthan, India

来源：

HETEROCYCLIC COMMUNICATIONS | 2010年 / 16卷 / 01期

关键词：

DERIVATIVES;

D O I：

10.1515/HC.2010.16.1.39

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Some new 4-[(substituted-benzothiazol-2-yl)-hydrazono]-2-(substituted phenyl) -5-methyl- 2, 4-dihydro-pyrazol-3-one (3) have been prepared by reacting substituted benzothiazol-2-yl amine with acetoacetic ester, 2-[substituted benzothiazol -2-yl)-hydrazono]-3-oxo-butyric acid ethyl ester (2) react with different hydrazines to give the title compounds. These compounds are evaluated for their antimicrobial activity. The structures of all these compounds have been confirmed by I.R., (1)HNMR,Mass spectra and elemental analysis data.

引用

页码：39 / 42

页数：4

共 50 条

[31] Synthesis and biological evaluation of novel 2-(substituted isoxazol-4-yl)-5-arylamino-1,3,4-oxadiazoles
Liu, Feng
Wang, Meiyan
Teng, Xinhuan
Zhang, Peizhi
Jiang, Lin
RESEARCH ON CHEMICAL INTERMEDIATES, 2014, 40 (04) : 1575 - 1581
[32] One-pot synthesis of 3-substituted-2-[(3-methyl-1H-pyrazol-5-yl)imino]-5,6-diphenyl-1,3-thiazin-4-ones
El-Sheref, Essmat M.
JOURNAL OF SULFUR CHEMISTRY, 2017, 38 (06) : 625 - 634
[33] SYNTHESIS AND ANTIULCER ACTIVITY OF NOVEL 2-[5-SUBSTITUTED 1H-BENZO (d) IMIDAZOLE-2-YL SULFINYL] METHYL 3-SUBSTITUTED QUINAZOLINE-4 (3H)-ONES
Patil, Avinash
Ganguly, Swastika
Surana, Sanjay
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2009, 19 (02) : 113 - 116
[34] Synthesis and in vitro antimicrobial screening of some 5-methyl-2-substituted phenyl-3-(phenylsulfonyl)thiazolidin-4-ones
Allahyani, Mamdouh
Almehmadi, Mazen
Abdulaziz, Osama
Alshamrani, Mohammed A.
Alzahrani, Abdullah Yahya Abdullah
Joshi, Kamal Kant
Asif, Mohammad
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2024, 34 (04) : 499 - 504
[35] Synthesis and Antimicrobial Screening of Some Novel 2-(5-(4-(1H-Benzo[d][1,2,3] triazol-1-yl)phenyl)-4,5-dihydro-1H-pyrazol3-yl) phenols Incorporated by Triazole Moiety
Shaikh, Mohammad U.
Jadhav, Ganesh R.
Kale, Rajesh P.
Chate, Asha V.
Nagargoje, Deepak R.
Gill, Charansingh H.
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2014, 51 (02) : 513 - 517
[36] Reactions of 2-(5-methyl-2-phenyl-2H-1,2,3-diazaphosphol-4-yl)-4H-1,3,2-benzodioxaphosphinin-4-one with chloral and hexafluoroacetone
Mironov, Vladimir F.
Ivkova, Gulnara A.
Abdrakhmanova, Liliya M.
Mironova, Ekaterina V.
Krivolapov, Dmitry B.
Konovalova, Irina V.
MENDELEEV COMMUNICATIONS, 2011, 21 (05) : 282 - 284
[37] Synthesis of methyl 2-[(1,2-dihydro-4-hydroxy-2-oxo-1-phenylquinolin-3-yl) carbonylamino] alkanoates and methyl 2-[2-(4,2-dihydro-4-hydroxy-2-oxo-1-phenylquinolin-3-ypcarbonyl-amino)alkanamido] alkanoate
Fathalla, Walid
Pazdera, Pavel
ARKIVOC, 2017, : 158 - 173
[38] Synthesis and antimicrobial screening of some 3-[4-(3-aryl-1-phenyl-1H-pyrazol-4-yl)-6-aryl-pyridin-2-yl] and 4-methyl-3-phenyl-6-[4-(3-aryl-1-phenyl-1H-pyrazol-4-yl)-6-aryl-pyridin-2-yl] coumarins
Brahmbhatt, D. I.
Kaneria, Ankit R.
Patel, Anil K.
Patel, Niraj H.
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 2010, 49 (07): : 971 - 977
[39] Synthesis, Antimicrobial Activity, Drug-likeness, and Molecular Docking Studies of Novel 3-((2-(Benzylthio)-5-(phenylselanyl) pyrimidin-4-yl)amino)-2-(4-substituted phenyl)thiazolidin-4-ones
Basha, N. Jeelan
Akshay, K. T.
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 2024, 56 (06) : 626 - 632
[40] 2-[3-(4-Methoxyphenyl)-1-phenyl-1H-pyrazol-5-yl]phenol
Kausar, Rukhsana
Badshah, Amir
ul Haq, Muhammad Zia
Hasan, Aurangzeb
Bolte, Michael
ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2009, 65 : O589 - U2416

← 1 2 3 4 5 →