Efficient One-Pot Synthesis of Benzimidazoles Under Solvent-Free Conditions

被引：23

作者：

Du, Li-Hua ^{[1
]}

Luo, Xi-Ping ^{[2
]}

机构：

[1] Zhejiang Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China

[2] Zhejiang Forestry Univ, Dept Environm Sci & Technol, Hangzhou, Zhejiang, Peoples R China

来源：

SYNTHETIC COMMUNICATIONS | 2010年 / 40卷 / 19期

关键词：

Benzimidazoles; green chemistry; iodobenzene diacetate (IBD); oxidations; INHIBITORS; BINDING; OXIDANT;

D O I：

10.1080/00397910903340629

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A green, efficient method for the synthesis of various 2-aryl-benzimidazoles in the presence of hypervalent iodine as the oxidant at room temperature under solvent-free conditions is reported. The salient features of this method include mild conditions, short reaction times (3-5min), excellent yields, and simple procedure.

引用

页码：2880 / 2886

页数：7

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