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- [33] Alzheimer's Disease-Rationales for Potential Treatment with the Thrombin Inhibitor DabigatranINTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (09)Grossmann, Klaus论文数: 0 引用数: 0 h-index: 0机构: Univ Tubingen, Ctr Plant Mol Biol ZMBP, D-72076 Tubingen, Germany Univ Tubingen, Ctr Plant Mol Biol ZMBP, D-72076 Tubingen, Germany
- [34] From Antipsychotic to Neuroprotective: Computational Repurposing of Fluspirilene as a Potential PDE5 Inhibitor for Alzheimer's DiseaseJOURNAL OF COMPUTATIONAL CHEMISTRY, 2025, 46 (02)Bhattacharya, Kunal论文数: 0 引用数: 0 h-index: 0机构: Assam Royal Global Univ, Royal Sch Pharm, Gauhati, India Pratiksha Inst Pharmaceut Sci, Dept Pharmaceut Chem, Gauhati, India Assam Royal Global Univ, Royal Sch Pharm, Gauhati, IndiaBhattacharjee, Atanu论文数: 0 引用数: 0 h-index: 0机构: Assam Royal Global Univ, Royal Sch Pharm, Gauhati, India Assam Royal Global Univ, Royal Sch Pharm, Gauhati, IndiaChakraborty, Manodeep论文数: 0 引用数: 0 h-index: 0机构: Himalayan Pharm Inst, Dept Pharmacol, Majhitar, India Assam Royal Global Univ, Royal Sch Pharm, Gauhati, IndiaDas, Dibyajyoti论文数: 0 引用数: 0 h-index: 0机构: Pratiksha Inst Pharmaceut Sci, Dept Pharmaceut Chem, Gauhati, India Dibrugarh Univ, Dept Pharmaceut Sci, Dibrugarh, India Assam Royal Global Univ, Royal Sch Pharm, Gauhati, IndiaPaudel, Keshav Raj论文数: 0 引用数: 0 h-index: 0机构: Centenary Inst, Ctr Inflammat, Sydney, NSW, Australia Univ Technol Sydney, Fac Sci, Sch Life Sci, Sydney, NSW, Australia Assam Royal Global Univ, Royal Sch Pharm, Gauhati, India
- [35] Design and optimization of heterocyclic 4-azaxanthenes as potent and selective inhibitors of BACE1 for the treatment of Alzheimer's diseaseABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Marx, Isaac E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAChen, Kui论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USACheng, Alan C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USADineen, Thomas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAEpstein, Oleg论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAEsmay, Joel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAHickman, Dean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAKreiman, Chuck E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWahl, Robert C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWen, Paul H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWeiss, Matthew M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWhittington, Douglas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWood, Stephen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAFremeau, Robert T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAWhite, Ryan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USAPatel, Vinod F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA Amgen Inc, Dept Med Chem, Cambridge, MA 02142 USA
- [36] Discovery of potent and selective dual cholinesterases and ?-secretase inhibitors in pomegranate as a treatment for Alzheimer?s diseaseBIOORGANIC CHEMISTRY, 2022, 129Ali, Md. Yousof论文数: 0 引用数: 0 h-index: 0机构: Univ Calgary, Hotchkiss Brain Inst, Cumming Sch Med, Dept Physiol & Pharmacol, Calgary, AB T2N 4N1, Canada Univ Calgary, Alberta Childrens Hosp Res Inst, Cumming Sch Med, Calgary, AB T2N 4N1, Canada Univ Calgary, Alberta Childrens Hosp Res Inst, Cumming Sch Med, Calgary, AB T2N 4N1, Canada Univ Calgary, Hotchkiss Brain Inst, Cumming Sch Med, Dept Physiol & Pharmacol, Calgary, AB T2N 4N1, CanadaZaib, Sumera论文数: 0 引用数: 0 h-index: 0机构: Univ Cent Punjab, Fac Life Sci, Dept Biochem, Lahore 54590, Pakistan Univ Calgary, Hotchkiss Brain Inst, Cumming Sch Med, Dept Physiol & Pharmacol, Calgary, AB T2N 4N1, CanadaJannat, Susoma论文数: 0 引用数: 0 h-index: 0机构: Univ Calgary, Dept Biochem & Mol Biol, Calgary, AB T2N 1N4, Canada Univ Calgary, Hotchkiss Brain Inst, Cumming Sch Med, Dept Physiol & Pharmacol, Calgary, AB T2N 4N1, CanadaKhan, Imtiaz论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Manchester Inst Biotechnol, 131 Princess St, Manchester M1 7DN, England Univ Calgary, Hotchkiss Brain Inst, Cumming Sch Med, Dept Physiol & Pharmacol, Calgary, AB T2N 4N1, Canada
- [37] Synthesis of Verubecestat, a BACE1 Inhibitor for the Treatment of Alzheimer's DiseaseORGANIC LETTERS, 2016, 18 (22) : 5780 - 5783Thaisrivongs, David K.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAMiller, Steven P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAMolinaro, Carmela论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAChen, Qinghao论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USASong, Zhiguo J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USATan, Lushi论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAChen, Lu论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Shanghai Pharmaceut Co Ltd, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAChen, Wenyong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USALekhal, Azzeddine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Engn Res & Dev, Proc Res & Dev, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAPulicare, Sarah K.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Engn Res & Dev, Proc Res & Dev, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USAXu, Yanke论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Engn Res & Dev, Proc Res & Dev, POB 2000, Rahway, NJ 07065 USA Merck Res Labs, Proc Chem, POB 2000, Rahway, NJ 07065 USA
- [38] Design, synthesis and biological evaluation of pyrazolopyrimidinone based potent and selective PDE5 inhibitors for treatment of erectile dysfunctionBIOORGANIC CHEMISTRY, 2019, 89Reddy, G. Lakshma论文数: 0 引用数: 0 h-index: 0机构: CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaDar, Mohd Ishaq论文数: 0 引用数: 0 h-index: 0机构: CSIR, Canc Pharmacol Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaHudwekar, Abhinandan D.论文数: 0 引用数: 0 h-index: 0机构: CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaMahajan, Priya论文数: 0 引用数: 0 h-index: 0机构: CSIR, Discovery Informat, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaNargotra, Amit论文数: 0 引用数: 0 h-index: 0机构: CSIR, Discovery Informat, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaBaba, Adil Manzoor论文数: 0 引用数: 0 h-index: 0机构: CSIR, Canc Pharmacol Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India CSIR, Pharmacol Div, Indian Inst Integrat Med, Srinagar 190005, Jammu & Kashmir, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaNandi, Utpal论文数: 0 引用数: 0 h-index: 0机构: CSIR, PK PD Tox Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaWazir, Priya论文数: 0 引用数: 0 h-index: 0机构: CSIR, PK PD Tox Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaSingh, Gurdarshan论文数: 0 引用数: 0 h-index: 0机构: CSIR, PK PD Tox Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaVishwakarma, Ram A.论文数: 0 引用数: 0 h-index: 0机构: CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaSyed, Sajad Hussain论文数: 0 引用数: 0 h-index: 0机构: CSIR, Canc Pharmacol Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Pharmacol Div, Indian Inst Integrat Med, Srinagar 190005, Jammu & Kashmir, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, IndiaSawant, Sanghapal D.论文数: 0 引用数: 0 h-index: 0机构: CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India Anusandhan Bhawan, Acad Sci & Innovat Res, 2 Rafi Marg, New Delhi 110001, India CSIR, Med Chem Div, Indian Inst Integrat Med, Canal Rd, Jammu 180001, Jammu & Kashmir, India
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