So what do we call GPR18 now?

被引：26

作者：

Alexander, S. P. H. ^{[1
]}

机构：

[1] Univ Nottingham, Sch Med, Sch Biomed Sci, Nottingham NG7 2UH, England

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 2012年 / 165卷 / 08期

关键词：

cannabinoid receptor; GPR18; anandamide; N-arachidonoylglycine; tetrahydrocannabinol; AM251; N-ARACHIDONOYL GLYCINE; IDENTIFICATION; ARACHIDONYLGLYCINE; LIGAND; ANANDAMIDE; INHIBITION;

D O I：

10.1111/j.1476-5381.2011.01731.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

The further characterization of the orphan GPCR GPR18 conducted by McHugh et al. in this issue of the British Journal of Pharmacology has generated a pharmacological profile that raises some interesting questions about the nomenclature of this receptor and may also prompt some questions about the pharmacological definition of the classical cannabinoid receptors, CB1 and CB2.

引用

页码：2411 / 2413

页数：3

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