Microwave assisted sulfopropylation of N-heterocycles using 1,3-propane sultone

被引：11

作者：

Adamczyk, M ^{[1
]}

Rege, S ^{[1
]}

机构：

[1] Abbott Labs, Div Organ Chem, Abbott Pk, IL 60064 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 52期

关键词：

D O I：

10.1016/S0040-4039(98)02301-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Dramatic rare acceleration was observed for N-sulfopropylation of heterocyclic compounds (1a-h) using 1,3-propane sultone(2) under microwave irradiation affording the N-sulfopropylated compounds (3a-h) in 68-95% yield. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：9587 / 9588

页数：2

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